SCHEMBL6680422

SCHEMBL6680422

CC(C)(C)OC(=O)NC1(c2cccc(N)c2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 2/20 0.39
CNR1 P21554 2/20 0.37
CNR2 P34972 2/20 0.37
GHSR Q92847 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ITGB1 P05556 1/20 0.35
ITGA4 P13612 1/20 0.35
ITGB7 P26010 1/20 0.35
AKT2 P31751 1/20 0.35
KIT P10721 1/20 0.35
NR1H2 P55055 2/20 0.34
ALOX15 P16050 2/20 0.34
TSHR P16473 1/20 0.34
ATM Q13315 1/20 0.34
CTSD P07339 2/20 0.34
BACE1 P56817 2/20 0.34
NR1H3 Q13133 1/20 0.33
DDX3X O00571 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6681079 0.95 AKT1 (0.37) AKT1CNR1CNR2GHSRHCRTR1
SCHEMBL6678166 0.95 AKT1 (0.39) AKT1CNR1CNR2GHSRHCRTR1
SCHEMBL6676765 0.94 SSTR4 (0.38) AKT1CNR1CNR2GHSRHCRTR1
SCHEMBL31360210 0.84 CTSB (0.40) AKT1CNR1CNR2ALDH1A1AKT2
SCHEMBL27425997 0.84 DRD2 (0.40) AKT1CNR1CNR2GHSRHCRTR1
SCHEMBL2036519 0.84 CTSB (0.40) AKT1CNR1CNR2ALDH1A1AKT2
SCHEMBL4087871 0.83 AKT1 (0.43) AKT1CNR1CNR2AKT2NR1H2
SCHEMBL2554955 0.83 AKT1 (0.47) AKT1CNR1CNR2ALDH1A1AKT2
SCHEMBL25155496 0.83 CNR1 (0.42) AKT1CNR1CNR2AKT2NR1H2
SCHEMBL30344050 0.83 CNR1 (0.42) AKT1CNR1CNR2AKT2NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
CN-1075808-C Aniline derivatives having nitric oxide synthase inhibitory activity CHUGAI PHARMACEUTICAL CO LTD (JP) 2001-12-05 CN disclosed
CN-1310169-A Anils with nitric oxide synzyme inhibiting function SHUGAI SEIYAKU K K (JP) 2001-08-29 CN disclosed
CN-1172473-A Aniline derivatives having nitric oxide synthase inhibitory activity CHUGAI PHARMACEUTICAL CO LTD (JP) 1998-02-04 CN disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed