SCHEMBL6680495

SCHEMBL6680495

CCN=C(N)Nc1ccccc1CCNC(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.47
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
NAMPT P43490 1/20 0.41
CACNA1C Q13936 1/20 0.41
SCN5A Q14524 1/20 0.41
LMNA P02545 2/20 0.40
POLB P06746 1/20 0.40
IDO1 P14902 4/20 0.40
MEN1 O00255 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
MALT1 Q9UDY8 1/20 0.38
NOS3 P29474 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6676657 0.78 CYP3A4 (0.47) NQO2GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7247902 0.76 NQO2 (0.46) NQO2NAMPTLMNAPOLBIDO1
SCHEMBL6674498 0.76 NQO2 (0.53) NQO2NAMPTLMNAPOLBIDO1
SCHEMBL31250995 0.75 NQO2 (0.56) NQO2NAMPTLMNAIDO1MEN1
SCHEMBL1231492 0.75 NQO2 (0.56) NQO2NAMPTLMNAIDO1MEN1
SCHEMBL6925241 0.75 NQO2 (0.56) NQO2SIGMAR1NAMPTLMNAIDO1
SCHEMBL6676329 0.75 SIGMAR1 (0.50) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6679750 0.74 NQO2 (0.50) NQO2NAMPTLMNAPOLBIDO1
SCHEMBL21680877 0.73 NQO2 (0.57) NQO2SIGMAR1NAMPTLMNAIDO1
SCHEMBL5757395 0.73 POLB (0.47) LMNAPOLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed