SCHEMBL6680680

SCHEMBL6680680

CCC(NC(=O)OC(C)(C)C)c1cccc(N)c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.43
CTSS P25774 1/20 0.43
CPN1 P15169 1/20 0.43
CPB2 Q96IY4 1/20 0.43
FAAH O00519 3/20 0.41
CA2 P00918 1/20 0.40
KLK5 Q9Y337 1/20 0.40
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39
ADRB3 P13945 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRB2 P47870 1/20 0.39
MAPT P10636 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SYK P43405 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16293719 0.87 CTSK (0.44) CTSKCTSSCPN1CPB2KLK5
SCHEMBL666640 0.87 CTSK (0.42) CTSKCTSSCPN1CPB2KLK5
SCHEMBL10311378 0.87 CTSK (0.44) CTSKCTSSCPN1CPB2KLK5
SCHEMBL27402040 0.86 KLK5 (0.43) CTSKCTSSKLK5MAPTALDH1A1
SCHEMBL5003031 0.86 TSHR (0.42) CTSKCTSSKLK5MAPTALDH1A1
SCHEMBL5003027 0.86 TSHR (0.42) CTSKCTSSKLK5MAPTALDH1A1
SCHEMBL665859 0.85 CTSK (0.41) CTSKCTSSCPN1CPB2KLK5
SCHEMBL6678205 0.83 FAAH (0.43) CTSKCTSSFAAHCA2ALDH1A1
SCHEMBL5212724 0.83 CTSK (0.56) CTSKCTSSFAAHMAPTALDH1A1
SCHEMBL12203909 0.83 CTSK (0.56) CTSKCTSSFAAHMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8871785-B2 Antiviral phosphonate analogs GILEAD SCIENCES, INC. (US) 2014-10-28 US disclosed
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed