SCHEMBL6680865

SCHEMBL6680865

O=C(Nc1ccccc1)c1cc(-c2ccccn2)cc(-n2ccccc2=O)c1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.46
KCNK3 O14649 1/20 0.45
KCNK9 Q9NPC2 1/20 0.45
F10 P00742 2/20 0.45
CYP2C9 P11712 2/20 0.45
NR4A2 P43354 1/20 0.45
CNR1 P21554 1/20 0.43
CYP3A4 P08684 1/20 0.43
ALDH1A1 P00352 1/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
RAB9A P51151 1/20 0.43
GFER P55789 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
PTPN2 P17706 1/20 0.43
PTPN1 P18031 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2763149 0.80 PTGS2 (0.43) F10CNR1LMNAPOLBSMN1; SMN2
SCHEMBL3667467 0.78 GRM5 (0.42) KDM4ELMNAPOLBRAB9A
SCHEMBL6689015 0.76 PRKDC (0.41) F10ALDH1A1KDM4ELMNAPOLB
SCHEMBL18074830 0.74 GRM5 (0.37) F10KDM4ELMNAPOLBRAB9A
SCHEMBL18573213 0.74 TRPV1 (0.71) TRPV1KCNK3KCNK9CNR1PTPN2
SCHEMBL14082180 0.74 TRPV1 (0.75) TRPV1KCNK3KCNK9POLBRAB9A
SCHEMBL31390061 0.73 KCNK3 (0.53) TRPV1KCNK3KCNK9CNR1PTPN2
SCHEMBL1881688 0.73 GRIA1 (0.51) TRPV1CYP2C9NR4A2CNR1CYP3A4
SCHEMBL3667668 0.72 GRM5 (0.53) F10ALDH1A1
SCHEMBL4372509 0.71 CHEK2 (0.41) F10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465626-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES Eisai Co., Ltd. (JP) 2004-10-13 EP disclosed
WO-2003047577-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES EISAI CO LTD (JP) 2003-06-12 WO disclosed