SCHEMBL6681071

SCHEMBL6681071

CC/N=C(/NC(=O)OC(C)(C)C)Nc1ccc(CCNC(=O)OC(C)(C)C)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.41
NAMPT P43490 1/20 0.38
IDO1 P14902 4/20 0.37
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
NR1H4 Q96RI1 1/20 0.37
PTPN11 Q06124 1/20 0.36
ITK Q08881 2/20 0.36
EGFR P00533 1/20 0.36
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
HPGD P15428 2/20 0.35
HTT P42858 2/20 0.35
KDM4E B2RXH2 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687607 0.89 IDO1 (0.44) NQO2NAMPTIDO1CA1CA2
SCHEMBL7243630 0.87 ALDH1A1 (0.42) NQO2NAMPTIDO1CA1CA2
SCHEMBL6681934 0.85 ALDH1A1 (0.42) NQO2NAMPTIDO1ALDH1A1GAA
SCHEMBL6681072 0.83 NQO2 (0.40) NQO2NAMPTIDO1CA1CA2
SCHEMBL6676112 0.83 NAMPT (0.54) NAMPTCA1CA2NR1H4PTPN11
SCHEMBL6688945 0.81 CYP3A4 (0.46) NQO2NAMPTIDO1CA1CA2
SCHEMBL6680791 0.80 NQO2 (0.44) NQO2NAMPTIDO1CA1CA2
SCHEMBL27493607 0.80 NQO2 (0.44) NQO2NAMPTIDO1CA1CA2
SCHEMBL7248116 0.80 CA1 (0.43) NQO2NAMPTCA1CA2MEN1
SCHEMBL6675303 0.79 NQO2 (0.40) NQO2ALDH1A1KMT2AKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed