SCHEMBL6688945

SCHEMBL6688945

CC/N=C(/NC(=O)OC(C)(C)C)Nc1cccc(CCNC(=O)OC(C)(C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.46
CYP2C19 P33261 2/20 0.46
AKT1 P31749 1/20 0.46
NAMPT P43490 1/20 0.44
CA2 P00918 3/20 0.43
CA1 P00915 2/20 0.43
NQO2 P16083 1/20 0.42
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
MAPK1 P28482 1/20 0.41
POLB P06746 2/20 0.40
HDAC6 Q9UBN7 1/20 0.39
CTSK P43235 1/20 0.39
NPFFR1 Q9GZQ6 3/20 0.39
NPFFR2 Q9Y5X5 3/20 0.39
IDO1 P14902 1/20 0.39
GLS O94925 1/20 0.38
NR1H4 Q96RI1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6676112 0.87 NAMPT (0.54) AKT1NAMPTCA2CA1CTSK
SCHEMBL6676657 0.86 CYP3A4 (0.47) CYP3A4CYP2C19AKT1NAMPTCA2
SCHEMBL6685803 0.86 ALDH1A1 (0.41) CYP3A4CYP2C19CA2CA1KDM4E
SCHEMBL6675938 0.84 CYP3A4 (0.47) CYP3A4CYP2C19AKT1NAMPTCA2
SCHEMBL6678215 0.84 PTGES (0.41) CYP3A4CYP2C19AKT1CA2CA1
SCHEMBL6687607 0.82 IDO1 (0.44) CYP3A4CYP2C19NAMPTCA2CA1
SCHEMBL6676258 0.82 CA1 (0.43) AKT1NAMPTCA2CA1NQO2
SCHEMBL6679114 0.82 SENP1 (0.48) MAPK1NPFFR1NPFFR2NR1H4
SCHEMBL7248116 0.81 CA1 (0.43) NAMPTCA2CA1NQO2
SCHEMBL7247586 0.81 CA1 (0.43) NAMPTCA2CA1NQO2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed