SCHEMBL6681752

SCHEMBL6681752

NC(=O)CCN1CCc2ccccc2C1=O

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.55
TSHR P16473 2/20 0.55
ALOX15 P16050 1/20 0.55
SIRT1 Q96EB6 1/20 0.55
BCAT2 O15382 1/20 0.50
DRD3 P35462 11/20 0.49
DRD1 P21728 5/20 0.49
DRD2 P14416 3/20 0.49
ACHE P22303 1/20 0.49
MEN1 O00255 1/20 0.49
POLB P06746 1/20 0.49
MAPT P10636 1/20 0.49
KMT2A Q03164 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
NPC1 O15118 1/20 0.47
ALDH1A1 P00352 1/20 0.47
RAB9A P51151 1/20 0.47
DRD4 P21917 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15690262 0.87 KDM4E (0.73) KDM4ETSHRALOX15SIRT1DRD3
SCHEMBL3785757 0.85 KDM4E (0.75) KDM4ETSHRALOX15SIRT1DRD3
SCHEMBL15690244 0.82 AOC3 (0.56) KDM4ETSHRALOX15SIRT1DRD3
SCHEMBL15691861 0.82 BCAT2 (0.47) KDM4ETSHRALOX15SIRT1BCAT2
SCHEMBL7149691 0.82 ITGB3 (0.51) MEN1KMT2A
SCHEMBL7686132 0.81 DRD3 (0.53) KDM4ETSHRALOX15SIRT1DRD3
SCHEMBL30183479 0.81 DRD3 (0.53) KDM4ETSHRALOX15SIRT1DRD3
SCHEMBL24169509 0.80 MAPT (0.74) KDM4ETSHRALOX15MEN1POLB
SCHEMBL11395534 0.80 CHRM2 (0.60) KDM4ETSHRALOX15SIRT1ACHE
SCHEMBL30183548 0.79 DRD3 (0.57) DRD3DRD1DRD2ACHEDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004004727-A1 3,4-DIHYDROISOQUINOLIN-1-ONE DERIVATIVES AS INDUCERS OF APOPTOSIS AXYS PHARMACEUTICALS, INC. (US) 2004-01-15 WO disclosed