SCHEMBL6681835

SCHEMBL6681835

CC/N=C(/NC(=O)OC(C)(C)C)Nc1ccc(NCc2ccccc2)c(CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.36
CA12 O43570 1/20 0.36
CA7 P43166 1/20 0.36
CA14 Q9ULX7 1/20 0.36
PTGES O14684 1/20 0.35
AKT1 P31749 2/20 0.35
HDAC1 Q13547 2/20 0.35
CA2 P00918 1/20 0.34
NPFFR1 Q9GZQ6 2/20 0.34
NPFFR2 Q9Y5X5 2/20 0.34
MAPKAPK2 P49137 1/20 0.34
ATM Q13315 1/20 0.34
AURKA O14965 2/20 0.34
RPS6KB1 P23443 2/20 0.34
NAMPT P43490 1/20 0.33
NR1H4 Q96RI1 1/20 0.33
MEN1 O00255 1/20 0.33
APAF1 O14727 1/20 0.33
KMT2A Q03164 1/20 0.33
SENP7 Q9BQF6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6681133 0.89 NR1H4 (0.34) CA1CA12MAPKAPK2NR1H4
SCHEMBL6679119 0.86 NR1H4 (0.35) CA1CA12CA2MAPKAPK2NR1H4
SCHEMBL6682103 0.86 AKT1 (0.37) PTGESAKT1HDAC1NPFFR1NPFFR2
SCHEMBL6679938 0.85 NR1H4 (0.36) CA1CA12CA2MAPKAPK2NR1H4
SCHEMBL6675974 0.84 CA1 (0.36) CA1CA12CA2MAPKAPK2NR1H4
SCHEMBL6678078 0.83 MAPKAPK2 (0.36) MAPKAPK2NR1H4MEN1KMT2A
SCHEMBL6675630 0.83 NR1H4 (0.35) CA1CA12MAPKAPK2NR1H4CTSK
SCHEMBL6681842 0.82 CA1 (0.34) CA1CA12CA7CA14HDAC1
SCHEMBL6675977 0.82 NR1H4 (0.35) CA1CA12CA2MAPKAPK2NR1H4
SCHEMBL6684393 0.81 NR1H4 (0.34) CA1CA12MAPKAPK2NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed