SCHEMBL6675974

SCHEMBL6675974

CC/N=C(/NC(=O)OC(C)(C)C)Nc1ccc(C)c(CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.36
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
MAPKAPK2 P49137 3/20 0.35
PTPN11 Q06124 1/20 0.34
CNR2 P34972 2/20 0.33
CYP17A1 P05093 1/20 0.33
GAA P10253 2/20 0.32
ALDH1A1 P00352 1/20 0.32
NR1I3 Q14994 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PSMB8 P28062 1/20 0.32
MCHR1 Q99705 1/20 0.32
BRD4 O60885 1/20 0.31
NPC1 O15118 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6679938 0.93 NR1H4 (0.36) CA1CA12CA9NR1H4MAPKAPK2
SCHEMBL6675630 0.91 NR1H4 (0.35) CA1CA12CA9NR1H4MAPKAPK2
SCHEMBL6678078 0.91 MAPKAPK2 (0.36) NR1H4MAPKAPK2PTPN11CYP17A1GAA
SCHEMBL6675977 0.90 NR1H4 (0.35) CA1CA12CA9NR1H4MAPKAPK2
SCHEMBL6679119 0.90 NR1H4 (0.35) CA1CA12CA9NR1H4MAPKAPK2
SCHEMBL6681133 0.89 NR1H4 (0.34) CA1CA12CA9NR1H4MAPKAPK2
SCHEMBL6684393 0.88 NR1H4 (0.34) CA1CA12CA9NR1H4MAPKAPK2
SCHEMBL6686106 0.87 NR1H4 (0.33) NR1H4MAPKAPK2PTPN11CYP17A1GAA
SCHEMBL6682277 0.86 KDM4E (0.39) NR1H4ALDH1A1NR1I3MEN1KMT2A
SCHEMBL6681835 0.84 CA1 (0.36) CA1CA12NR1H4MAPKAPK2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed