SCHEMBL6681863

SCHEMBL6681863

Cc1cc(N)cc(CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.39
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
HDAC8 Q9BY41 1/20 0.34
PARP10 Q53GL7 1/20 0.33
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
TSPO P30536 2/20 0.31
AAK1 Q2M2I8 1/20 0.30
HTR2C P28335 1/20 0.30
SLC6A4 P31645 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
NCOR2 Q9Y618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4535348 0.85 HDAC1 (0.37) ALDH1A1TSHRHDAC8NFKB1NFKB2
SCHEMBL4530344 0.83 AAK1 (0.34) ALDH1A1TSHRHDAC8PARP10TSPO
SCHEMBL6678261 0.82 CETP (0.43) GRM2
SCHEMBL1099618 0.81 CETP (0.39) HDAC8NFKB1NFKB2RELAHDAC3
SCHEMBL7247305 0.79 GRM2 (0.43) GRM2HTR2CSLC6A4HDAC3HDAC1
SCHEMBL6680561 0.79 GRM2 (0.37) GRM2
SCHEMBL7944783 0.78 GRM2 (0.44) GRM2NFKB1HDAC3HDAC1HDAC2
SCHEMBL6679733 0.78 TSHR (0.44) GRM2ALDH1A1TSHR
SCHEMBL27389057 0.78 ALDH1A1 (0.43) ALDH1A1TSHRPARP10TSPOHDAC1
SCHEMBL6680557 0.78 CYP1A2 (0.38) GRM2ALDH1A1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed