SCHEMBL6682277

SCHEMBL6682277

CC/N=C(/NC(=O)OC(C)(C)C)Nc1ccc(N2CCCC2)c(CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
RECQL P46063 1/20 0.39
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C19 P33261 1/20 0.36
NR1I3 Q14994 3/20 0.36
ALDH1A1 P00352 4/20 0.35
ACHE P22303 2/20 0.35
BACE1 P56817 2/20 0.35
NPSR1 Q6W5P4 3/20 0.35
NR1H4 Q96RI1 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
MAPT P10636 1/20 0.33
NPC1 O15118 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6679938 0.87 NR1H4 (0.36) NR1I3ALDH1A1NR1H4
SCHEMBL6675974 0.86 CA1 (0.36) MEN1KMT2ACYP2C19NR1I3ALDH1A1
SCHEMBL6675630 0.85 NR1H4 (0.35) NR1I3ALDH1A1NR1H4NPC1HPGD
SCHEMBL6678078 0.85 MAPKAPK2 (0.36) MEN1KMT2ACYP2D6CYP2C19ALDH1A1
SCHEMBL6679310 0.85 KDM4E (0.40) KDM4ERECQLMEN1KMT2ACYP2D6
SCHEMBL6675977 0.85 NR1H4 (0.35) KMT2ANR1I3ALDH1A1NR1H4HPGD
SCHEMBL6679119 0.85 NR1H4 (0.35) NR1I3ALDH1A1NR1H4
SCHEMBL6681133 0.84 NR1H4 (0.34) NR1I3ALDH1A1NR1H4
SCHEMBL6684393 0.83 NR1H4 (0.34) KDM4ENR1I3ALDH1A1NR1H4MAPT
SCHEMBL6686106 0.82 NR1H4 (0.33) NR1I3ALDH1A1NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed