SCHEMBL6682503

SCHEMBL6682503

COC(=O)CCc1cc(Br)c(O)c(C=O)c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 7/20 0.47
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
IDO1 P14902 1/20 0.36
ALOX5 P09917 1/20 0.36
EGFR P00533 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
PTPN1 P18031 1/20 0.35
HSP90AB1 P08238 1/20 0.35
PRKDC P78527 1/20 0.35
GAA P10253 1/20 0.35
THRA P10827 3/20 0.35
THRB P10828 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3130670 0.86 TRPV1 (0.44) LMNAMAPTIDO1ALOX5TRPV1
SCHEMBL1302419 0.85 HSP90AB1 (0.51) ERN1LMNAMAPTHSP90AB1PRKDC
SCHEMBL5072092 0.79 TRPV1 (0.54) MAPTALOX5TRPV1PTPN1GAA
SCHEMBL3679438 0.79 RPS6KA3 (0.39) MAPTIDO1ALOX5TRPV1PTPN1
SCHEMBL3684924 0.79 THRA (0.39) MAPTIDO1ALOX5TRPV1HSP90AB1
SCHEMBL4930870 0.77 TSHR (0.45) TRPV1PTPN1HSP90AB1THRATHRB
SCHEMBL30185945 0.77 CDK1 (0.59) ERN1ALOX5PTPN1GAA
SCHEMBL15543678 0.77 CDK1 (0.59) ERN1ALOX5PTPN1GAA
SCHEMBL18232227 0.76 PTPN1 (0.43) LMNAMAPTIDO1ALOX5PTPN1
SCHEMBL28131968 0.76 TRPV1 (0.47) LMNATRPV1HSP90AB1THRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004062661-A1 2-‘5-(5-CARBAMIMIDOYL-1H-HETEROARYL)-6-HYDROXYBIPHENYL-3-YL!- CARBOXYLIC ACID DERIVATIVES AS FACTOR VIIA INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2004-07-29 WO disclosed