SCHEMBL6684550

SCHEMBL6684550

NC(=O)COc1ccc2c(c1)S(=O)(=O)N=C(c1c(O)c3ccccc3n(CCC3CC3)c1=O)N2

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.82
NR1I2 O75469 1/20 0.61
MAPK1 P28482 1/20 0.49
HSD17B10 Q99714 1/20 0.49
HIF1A Q16665 1/20 0.38
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
PARP1 P09874 1/20 0.32
PARP2 Q9UGN5 1/20 0.32
DPP4 P27487 4/20 0.32
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
GAA P10253 1/20 0.32
PTGER4 P35408 1/20 0.32
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
ADORA1 P30542 1/20 0.31
PSEN1 P49768 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6267035 0.94 CYP2C9 (0.90) CYP2C9NR1I2MAPK1HSD17B10HIF1A
SCHEMBL6234512 0.90 CYP2C9 (1.00) CYP2C9NR1I2MAPK1HSD17B10HIF1A
SCHEMBL6736116 0.90 CYP2C9 (0.84) CYP2C9NR1I2MAPK1HSD17B10HIF1A
SCHEMBL7075766 0.90 CYP2C9 (0.73) CYP2C9NR1I2MAPK1HSD17B10HIF1A
SCHEMBL6692151 0.89 CYP2C9 (0.67) CYP2C9NR1I2MAPK1HSD17B10HIF1A
SCHEMBL6681450 0.89 CYP2C9 (0.66) CYP2C9NR1I2MAPK1HSD17B10KDM4E
SCHEMBL6738292 0.88 CYP2C9 (0.65) CYP2C9NR1I2MAPK1HSD17B10HIF1A
SCHEMBL6239158 0.87 CYP2C9 (0.63) CYP2C9NR1I2MAPK1HSD17B10KDM4E
SCHEMBL1522252 0.87 CYP2C9 (0.63) CYP2C9NR1I2MAPK1HSD17B10KDM4E
SCHEMBL1522640 0.86 CYP2C9 (0.61) CYP2C9NR1I2MAPK1HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004052312-A2 ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2004-06-24 WO claimed