SCHEMBL6692151

SCHEMBL6692151

NC(=O)COc1ccc2c(c1)S(=O)(=O)N=C(c1c(O)c3ccccc3n(CC3CCC3)c1=O)N2

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.67
MAPK1 P28482 1/20 0.49
HSD17B10 Q99714 1/20 0.49
NR1I2 O75469 1/20 0.48
NPC1 O15118 1/20 0.40
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
HIF1A Q16665 1/20 0.35
GSK3B P49841 1/20 0.34
EGLN1 Q9GZT9 5/20 0.34
PLA2G2A P14555 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6736069 0.90 CYP2C9 (0.82) CYP2C9MAPK1HSD17B10NR1I2NPC1
SCHEMBL6684550 0.89 CYP2C9 (0.82) CYP2C9MAPK1HSD17B10NR1I2HIF1A
SCHEMBL1522398 0.87 CYP2C9 (0.59) CYP2C9MAPK1HSD17B10NR1I2NPC1
SCHEMBL1522640 0.86 CYP2C9 (0.61) CYP2C9MAPK1HSD17B10NR1I2NPC1
SCHEMBL6685735 0.85 MAPK1 (0.57) CYP2C9MAPK1HSD17B10NR1I2NPC1
SCHEMBL1522203 0.85 CYP2C9 (0.59) CYP2C9MAPK1HSD17B10NR1I2NPC1
SCHEMBL1522252 0.85 CYP2C9 (0.63) CYP2C9MAPK1HSD17B10NR1I2KDM4E
SCHEMBL6681450 0.85 CYP2C9 (0.66) CYP2C9MAPK1HSD17B10NR1I2KDM4E
SCHEMBL1522450 0.84 CYP2C9 (0.59) CYP2C9MAPK1HSD17B10NR1I2NPC1
SCHEMBL6239158 0.84 CYP2C9 (0.63) CYP2C9MAPK1HSD17B10NR1I2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004052312-A2 ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2004-06-24 WO claimed