SCHEMBL6681450

SCHEMBL6681450

CC(C)(C)CCn1c(=O)c(C2=NS(=O)(=O)c3cc(OCC(N)=O)ccc3N2)c(O)c2ccccc21

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.66
MAPK1 P28482 1/20 0.53
HSD17B10 Q99714 1/20 0.53
NR1I2 O75469 1/20 0.47
DPP4 P27487 4/20 0.36
KDM4E B2RXH2 5/20 0.34
GAA P10253 2/20 0.34
ALDH1A1 P00352 4/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6692294 0.91 CYP2C9 (0.80) CYP2C9MAPK1HSD17B10NR1I2DPP4
SCHEMBL6239158 0.90 CYP2C9 (0.63) CYP2C9MAPK1HSD17B10NR1I2DPP4
SCHEMBL6684550 0.89 CYP2C9 (0.82) CYP2C9MAPK1HSD17B10NR1I2DPP4
SCHEMBL1522640 0.87 CYP2C9 (0.61) CYP2C9MAPK1HSD17B10NR1I2DPP4
SCHEMBL6686456 0.85 HSD17B10 (0.61) CYP2C9MAPK1HSD17B10NR1I2KDM4E
SCHEMBL6692151 0.85 CYP2C9 (0.67) CYP2C9MAPK1HSD17B10NR1I2KDM4E
SCHEMBL6231859 0.83 CYP2C9 (0.69) CYP2C9MAPK1HSD17B10NR1I2DPP4
SCHEMBL1380681 0.83 CYP2C9 (0.55) CYP2C9MAPK1HSD17B10NR1I2DPP4
SCHEMBL6235373 0.83 HSD17B10 (0.74) CYP2C9MAPK1HSD17B10NR1I2KDM4E
SCHEMBL6235277 0.83 MAPK1 (0.59) CYP2C9MAPK1HSD17B10NR1I2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004052312-A2 ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2004-06-24 WO claimed
WO-2004052312-A2 ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2004-06-24 WO disclosed