SCHEMBL6686671

SCHEMBL6686671

COc1ccc(F)cc1C(C)(C)CC(O)(C(=O)Nc1ccccc1)C(F)(F)F

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 19/20 0.68
PGR P06401 5/20 0.68
NR3C2 P08235 10/20 0.64
AR P10275 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6686666 0.86 NR3C1 (0.67) NR3C1PGRNR3C2AR
SCHEMBL1775018 0.84 NR3C1 (0.67) NR3C1PGRNR3C2
SCHEMBL1775956 0.84 NR3C1 (0.67) NR3C1PGRNR3C2
SCHEMBL1775343 0.84 NR3C1 (0.67) NR3C1PGRNR3C2
SCHEMBL4617886 0.83 NR3C1 (0.72) NR3C1PGRNR3C2
SCHEMBL4817160 0.82 NR3C2 (0.61) NR3C1PGRNR3C2
SCHEMBL6585107 0.82 NR3C1 (1.00) NR3C1PGRNR3C2AR
SCHEMBL5517620 0.79 NR3C2 (0.65) NR3C1PGRNR3C2
SCHEMBL4618245 0.79 NR3C1 (0.57) NR3C1PGRNR3C2AR
SCHEMBL6685141 0.79 NR3C1 (0.55) NR3C1PGRNR3C2AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040224992-A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2004-11-11 US claimed
WO-2004075864-A2 GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2004-09-10 WO claimed
US-20040224992-A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2004-11-11 US disclosed
WO-2004075864-A2 GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2004-09-10 WO disclosed
WO-2004046826-A2 POSITIVE TONE LITHOGRAPHY IN CARBON DIOXIDE SOLVENTS MICELL TECHNOLOGIES, INC. (US) 2004-06-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040224992-A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof NR3C1, NR3C2, MC2R NR3C1 1/4885PGR 173/4885NR3C2 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.