SCHEMBL6687282

SCHEMBL6687282

COc1ccc(-n2nc(C(F)(F)F)nc2-c2ccc(OCCCNC(N)=O)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.53
PTGS1 P23219 4/20 0.53
L3MBTL1 Q9Y468 1/20 0.50
MALT1 Q9UDY8 2/20 0.47
CYP3A4 P08684 3/20 0.43
CYP2C9 P11712 3/20 0.43
CYP2C19 P33261 1/20 0.43
MYOF Q9NZM1 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2B6 P20813 2/20 0.42
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA7 P43166 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687455 0.90 PTGS2 (0.42) PTGS2PTGS1L3MBTL1MALT1CYP3A4
SCHEMBL6687179 0.89 PTGS2 (0.71) PTGS2PTGS1L3MBTL1MALT1CYP3A4
SCHEMBL6681028 0.87 PTGS2 (0.53) PTGS2PTGS1L3MBTL1MALT1
SCHEMBL6682106 0.84 PTGS2 (0.60) PTGS2PTGS1L3MBTL1MALT1CYP3A4
Hydrochloric Acid SCHEMBL6687629 0.83 PTGS2 (0.58) PTGS2PTGS1L3MBTL1MALT1CYP3A4
SCHEMBL6682132 0.83 PTGS2 (0.53) PTGS2PTGS1L3MBTL1MALT1
SCHEMBL5148697 0.81 PTGS2 (0.46) PTGS2PTGS1L3MBTL1MALT1MTNR1A
SCHEMBL6132473 0.80 PTGS2 (0.67) PTGS2PTGS1L3MBTL1CYP3A4CYP2C9
SCHEMBL6686281 0.80 MALT1 (0.54) PTGS2PTGS1L3MBTL1MALT1MTNR1A
SCHEMBL5147861 0.80 PTGS2 (0.65) PTGS2PTGS1CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004060367-A1 IMIDAZOLE AND TRIAZOLE DERIVATIVES USEFUL AS SELECTIVE COX-1 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-07-22 WO disclosed