SCHEMBL6687535

SCHEMBL6687535

COc1cc(OCc2ccc(SC(F)(F)F)cc2)ccc1CNC(Cc1ccccc1)C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.44
ITGB7 P26010 1/20 0.44
CD274 Q9NZQ7 4/20 0.44
PPARG P37231 2/20 0.43
PPARA Q07869 2/20 0.43
FFAR1 O14842 1/20 0.43
PPARD Q03181 1/20 0.42
PTPRZ1 P23471 1/20 0.42
PDCD1 Q15116 2/20 0.41
MAOB P27338 3/20 0.41
FFAR4 Q5NUL3 1/20 0.41
MAOA P21397 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687567 0.90 PPARG (0.42) ITGA4ITGB7CD274PPARGPTPRZ1
SCHEMBL6687562 0.90 PPARG (0.42) ITGA4ITGB7CD274PPARGPTPRZ1
SCHEMBL6689339 0.88 PTPRZ1 (0.43) CD274PPARGPPARAPPARDPTPRZ1
SCHEMBL6689649 0.88 MAOB (0.51) PPARGPTPRZ1MAOBMAOA
SCHEMBL6687537 0.88 PTPRZ1 (0.43) CD274PPARGPPARAPPARDPTPRZ1
SCHEMBL6688970 0.86 MAOB (0.52) CD274PPARAPTPRZ1MAOBMAOA
SCHEMBL6690781 0.86 MAOB (0.52) CD274PPARAPTPRZ1MAOBMAOA
SCHEMBL6691341 0.86 PTPRZ1 (0.53) PPARGPTPRZ1MAOBMAOA
SCHEMBL6685530 0.81 FFAR4 (0.48) CD274PPARGPPARAFFAR1FFAR4
SCHEMBL6685527 0.81 FFAR4 (0.48) CD274PPARGPPARAFFAR1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed