SCHEMBL6687945

SCHEMBL6687945

COC(=O)c1ccc(OCc2c(F)cccc2F)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.58
RAB9A P51151 6/20 0.56
KMT2A Q03164 3/20 0.55
ALDH1A1 P00352 1/20 0.55
NPC1 O15118 5/20 0.54
SMN1; SMN2 Q16637 5/20 0.54
MEN1 O00255 2/20 0.54
MAOB P27338 2/20 0.51
MRGPRX4 Q96LA9 2/20 0.51
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
NR1H4 Q96RI1 1/20 0.50
POLB P06746 1/20 0.50
BLM P54132 1/20 0.50
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
PARP15 Q460N3 1/20 0.48
PARP14 Q460N5 1/20 0.48
PARP10 Q53GL7 1/20 0.48
CA12 O43570 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10395976 0.90 NR1H4 (0.56) MAPTRAB9AKMT2AALDH1A1NPC1
SCHEMBL2088021 0.85 ALDH1A1 (0.59) MAPTRAB9AKMT2AALDH1A1NPC1
SCHEMBL2087289 0.84 MAOB (0.70) ALDH1A1SMN1; SMN2MAOBL3MBTL1
SCHEMBL1444069 0.84 MAOB (0.74) MAPTRAB9AKMT2AALDH1A1NPC1
SCHEMBL2087038 0.83 NR4A2 (0.61) RAB9ANPC1SMN1; SMN2MAOBPOLB
SCHEMBL10396460 0.82 NR1H4 (0.62) MAPTRAB9AKMT2ANPC1SMN1; SMN2
SCHEMBL31530400 0.81 CA12 (0.50) MAPTRAB9AKMT2AALDH1A1NPC1
SCHEMBL11348928 0.80 MAPT (0.64) MAPTRAB9AKMT2ANPC1SMN1; SMN2
SCHEMBL11349807 0.80 MAPT (0.64) MAPTRAB9AKMT2ANPC1SMN1; SMN2
SCHEMBL2090015 0.79 GSK3B (0.50) RAB9ANPC1SMN1; SMN2MAOBPARP15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed