SCHEMBL6689108

SCHEMBL6689108

CC(=O)C(c1cccnc1)C1CCOCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.46
HSD17B10 Q99714 1/20 0.46
FPR2 P25090 1/20 0.42
CYP2C9 P11712 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 1/20 0.41
P2RX7 Q99572 1/20 0.40
NAMPT P43490 1/20 0.40
MAPT P10636 2/20 0.40
CYP3A5 P20815 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
THRB P10828 1/20 0.40
KCNA5 P22460 1/20 0.40
POLB P06746 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
CYP17A1 P05093 2/20 0.39
CYP19A1 P11511 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17065013 0.90 CYP3A4 (0.44) ALDH1A1HSD17B10CYP2C9CYP3A4CYP2C19
SCHEMBL6687691 0.84 ALDH1A1 (0.39) ALDH1A1KDM4EHSD17B10FPR2CYP2C9
SCHEMBL29062262 0.83 ALDH1A1 (0.47) ALDH1A1KDM4EHSD17B10P2RX7MAPT
SCHEMBL28143235 0.79 TP53 (0.53) ALDH1A1MAPTRAB9ASMN1; SMN2THRB
SCHEMBL2425571 0.78 SMN1; SMN2 (0.46) ALDH1A1KDM4EHSD17B10FPR2CYP2C9
SCHEMBL14428532 0.77 ALDH1A1 (0.43) ALDH1A1KDM4EHSD17B10CYP2C9CYP3A4
SCHEMBL5378828 0.76 SLC6A4 (0.42) ALDH1A1KDM4EHSD17B10FPR2CYP3A4
SCHEMBL12282165 0.74 SLC6A4 (0.45) ALDH1A1KDM4EHSD17B10
SCHEMBL29587838 0.73 ALDH1A1 (0.39) ALDH1A1KDM4EHSD17B10CYP2C9CYP3A4
SCHEMBL28144222 0.73 RAB9A (0.58) ALDH1A1KDM4EHSD17B10CYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004108668-A2 ALPHA-7 NEURONAL NICOTINIC RECEPTOR LIGANDS: COMPOSITIONS AND METHODS OF USE TARGACEPT, INC. (US) 2004-12-16 WO disclosed
EP-0994875-A1 3-PYRIDYL-1-AZA-BICYCLO-ALKANE DERIVATIVES FOR PREVENTION AND TREATMENT OF CNS DISORDERS R.J. REYNOLDS TOBACCO COMPANY (US) 2000-04-26 EP disclosed
WO-1999000385-A1 3-PYRIDYL-1-AZA-BICYCLO-ALKANE DERIVATIVES FOR PREVENTION AND TREATMENT OF CNS DISORDERS R.J. REYNOLDS TOBACCO COMPANY (US) 1999-01-07 WO disclosed