SCHEMBL6689959

SCHEMBL6689959

NC(=O)Cc1ccccc1OCCCN(CC(c1ccccc1)C1CCCCC1)C1CCN(C(=O)c2ccccc2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
EPHX2 P34913 1/20 0.36
PARP1 P09874 2/20 0.35
CYP3A4 P08684 2/20 0.34
DRD3 P35462 2/20 0.34
CHRM2 P08172 1/20 0.34
HTR1A P08908 1/20 0.34
ADRA2A P08913 1/20 0.34
CHRM1 P11229 1/20 0.34
DRD1 P21728 1/20 0.34
SLC6A2 P23975 1/20 0.34
ADRA1A P35348 1/20 0.34
OPRM1 P35372 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KCNH2 Q12809 1/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6698166 0.91 MEN1 (0.38) MEN1KMT2ACYP3A4DRD3CHRM2
SCHEMBL6515535 0.86 NR1H3 (0.46) MEN1KMT2ALMNAKDM4EALDH1A1
SCHEMBL6515170 0.84 NR1H3 (0.44) MEN1KMT2AOPRM1KCNH2HRH3
SCHEMBL7073248 0.80 LMNA (0.40) MEN1KMT2ALMNAPOLBALDH1A1
SCHEMBL6515545 0.78 NR1H3 (0.44) MEN1KMT2AOPRM1KCNH2HRH3
SCHEMBL6510586 0.77 NR1H3 (0.48) MEN1KMT2AALDH1A1HRH3
SCHEMBL6512055 0.77 NR1H3 (0.45) MEN1KMT2AOPRM1KCNH2LMNA
SCHEMBL6513610 0.76 NR1H3 (0.45) MEN1KMT2ALMNAKDM4EALDH1A1
SCHEMBL6519456 0.75 NR1H3 (0.43) CYP3A4DRD3CHRM2HTR1AADRA2A
SCHEMBL6515146 0.74 NR1H3 (0.55) MEN1KMT2ALMNAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2004509161-A 2004-03-25 JP claimed
EP-1318976-A2 SUBSTITUTED AMINOPROPOXYARYL DERIVATIVES USEFUL AS AGONISTS FOR LXR GLAXO GROUP LIMITED (GB) 2003-06-18 EP claimed
WO-2002024632-A2 SUBSTITUTED AMINOPROPOXYARYL DERIVATIVES USEFUL AS AGONISTS FOR LXR GLAXO GROUP LIMITED (GB) 2002-03-28 WO claimed