SCHEMBL6690125

SCHEMBL6690125

CS(=O)(=O)Nc1cccc(C(=O)NCC(C(=O)NCCNc2ccc(F)cc2)C2CCCCC2)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 2/20 0.49
CTSS P25774 8/20 0.47
CTSL P07711 7/20 0.47
CTSK P43235 4/20 0.47
HTR2B P41595 1/20 0.46
ALDH1A1 P00352 2/20 0.41
KMT2A Q03164 1/20 0.41
ANO1 Q5XXA6 1/20 0.41
MAPK14 Q16539 1/20 0.40
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PKM P14618 1/20 0.39
EPHX2 P34913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6690045 0.90 ALDH1A1 (0.51) CTSSCTSLCTSKALDH1A1KMT2A
SCHEMBL6688308 0.89 CTSS (0.47) CTSSCTSLCTSKHTR2BALDH1A1
SCHEMBL6687888 0.83 EPHX2 (0.51) CTSSCTSLCTSKKMT2AEPHX2
SCHEMBL6688266 0.82 HTR2B (0.47) CTSSCTSLCTSKHTR2BALDH1A1
SCHEMBL5843145 0.82 CTSS (0.63) CTSSCTSLCTSK
SCHEMBL5843139 0.82 CTSS (0.63) CTSSCTSLCTSK
SCHEMBL6692456 0.77 CTSS (0.62) CTSSCTSLCTSK
SCHEMBL6687973 0.77 EPHX2 (0.50) CTSSCTSLCTSKKMT2AEPHX2
SCHEMBL6687678 0.76 CTSS (0.71) CTSSCTSLCTSKPKM
SCHEMBL6690860 0.76 CTSS (0.61) CTSSCTSLCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084842-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed