SCHEMBL6690939

SCHEMBL6690939

COC(=O)CC(NC(=O)CNC(=O)OCc1ccccc1)c1ccc(O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.49
TSHR P16473 1/20 0.48
MAPT P10636 1/20 0.48
NPBWR1 P48145 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MCHR1 Q99705 1/20 0.48
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
HTT P42858 1/20 0.47
MAPK1 P28482 1/20 0.47
KLK1 P06870 1/20 0.46
CASP1 P29466 1/20 0.43
CTSL P07711 2/20 0.42
CTSS P25774 2/20 0.42
CTSB P07858 1/20 0.42
CTSK P43235 1/20 0.42
LMNA P02545 1/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7304322 0.85 CYP3A4 (0.53) CYP3A4TSHRMAPTNPBWR1NPSR1
SCHEMBL7146807 0.83 CYP3A4 (0.54) CYP3A4TSHRALDH1A1SMN1; SMN2HTT
SCHEMBL16201457 0.82 ATM (0.54) CYP3A4TSHRALDH1A1SMN1; SMN2MAPK1
SCHEMBL6958944 0.82 ATM (0.54) CYP3A4TSHRALDH1A1SMN1; SMN2MAPK1
SCHEMBL9683154 0.81 MAPT (0.51) CYP3A4TSHRMAPTNPBWR1NPSR1
SCHEMBL5700948 0.79 F2 (0.49) CYP3A4TSHRALDH1A1CASP1CTSL
SCHEMBL5700951 0.79 F2 (0.49) CYP3A4TSHRALDH1A1CASP1CTSL
SCHEMBL13588071 0.77 MDM4 (0.61) TSHRALDH1A1CTSLCTSSCTSB
SCHEMBL28902023 0.77 MDM4 (0.61) TSHRALDH1A1CTSLCTSSCTSB
SCHEMBL14501542 0.77 MAPK1 (0.55) CYP3A4TSHRMAPTNPBWR1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004091542-A2 NITROGEN CONTAINING INTEGRIN TARGETING COMPOUNDS COVX PHARMACEUTICALS, INC. (US) 2004-10-28 WO disclosed