SCHEMBL9683154

SCHEMBL9683154

COC(=O)C[C@H](NC(=O)CNC(=O)OCc1ccccc1)C(=O)OC

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.51
NPBWR1 P48145 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
MCHR1 Q99705 1/20 0.51
ALDH1A1 P00352 3/20 0.50
CYP3A4 P08684 2/20 0.50
MAPK1 P28482 1/20 0.50
KDM4E B2RXH2 1/20 0.50
GAA P10253 1/20 0.50
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
KYNU Q16719 1/20 0.49
TSHR P16473 1/20 0.48
CASP1 P29466 1/20 0.47
ALOX15 P16050 1/20 0.47
ATM Q13315 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19327506 0.90 KLK5 (0.51) MAPTNPBWR1NPSR1MCHR1ALDH1A1
SCHEMBL19327507 0.90 KLK5 (0.51) MAPTNPBWR1NPSR1MCHR1ALDH1A1
SCHEMBL31377319 0.88 MAPT (0.49) MAPTNPBWR1NPSR1MCHR1ALDH1A1
SCHEMBL22811132 0.88 MAPK1 (0.52) MAPTNPBWR1NPSR1MCHR1ALDH1A1
SCHEMBL8932374 0.88 MAPK1 (0.52) MAPTNPBWR1NPSR1MCHR1ALDH1A1
SCHEMBL9491221 0.88 ATM (0.59) ALDH1A1CYP3A4TSHRALOX15ATM
SCHEMBL330432 0.88 ATM (0.59) ALDH1A1CYP3A4TSHRALOX15ATM
SCHEMBL12400686 0.87 KYNU (0.62) ALDH1A1KYNUCASP1ALOX15
SCHEMBL2617394 0.87 KYNU (0.62) ALDH1A1KYNUCASP1ALOX15
SCHEMBL8932361 0.86 MAPK1 (0.51) MAPTNPBWR1NPSR1MCHR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5144073-A Decyclization of diketopiperazine intermediates EASTMAN CHEMICAL COMPANY 1992-09-01 US disclosed