SCHEMBL6690944

SCHEMBL6690944

COc1cc(OCc2c(F)cccc2Cl)ccc1CNC(Cc1ccccc1)C(N)=O

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.48
MAOA P21397 1/20 0.48
CD274 Q9NZQ7 2/20 0.46
FFAR1 O14842 2/20 0.45
ITGA4 P13612 5/20 0.43
PARP15 Q460N3 1/20 0.43
PARP10 Q53GL7 1/20 0.43
TP53 P04637 1/20 0.43
ITGB1 P05556 1/20 0.43
LMNA P02545 1/20 0.43
STING1 Q86WV6 1/20 0.42
ITGB7 P26010 1/20 0.42
FFAR4 Q5NUL3 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
EGFR P00533 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687864 0.94 MAOB (0.45) MAOBMAOACD274FFAR1ITGA4
SCHEMBL6687860 0.94 MAOB (0.45) MAOBMAOACD274FFAR1ITGA4
SCHEMBL6685101 0.91 CD274 (0.45) CD274ITGA4TP53ITGB1LMNA
SCHEMBL6685099 0.91 CD274 (0.45) CD274ITGA4TP53ITGB1LMNA
SCHEMBL6685482 0.88 MAOB (0.47) MAOBMAOACD274PARP15PARP10
SCHEMBL6685476 0.88 MAOB (0.47) MAOBMAOACD274PARP15PARP10
SCHEMBL6687664 0.86 MAOB (0.59) MAOBMAOACD274PARP15PARP10
SCHEMBL6687667 0.86 MAOB (0.59) MAOBMAOACD274PARP15PARP10
SCHEMBL6691050 0.85 KMT2A (0.43) MAOBMAOACD274ITGA4ITGB1
SCHEMBL6691044 0.85 KMT2A (0.43) MAOBMAOACD274ITGA4ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed