SCHEMBL6691028

SCHEMBL6691028

CNC(=O)[C@@H](NCc1ccc(OCc2cc(CF)cc(CF)c2)cc1)C(C)O

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.46
SCN9A Q15858 2/20 0.46
MAOA P21397 1/20 0.46
PDCD1 Q15116 2/20 0.40
CD274 Q9NZQ7 2/20 0.40
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
BCHE P06276 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6691022 1.00 MAOB (0.46) MAOBSCN9AMAOAPDCD1CD274
SCHEMBL3288931 0.86 BCHE (0.55) MEN1POLBMAPK1KMT2ANPSR1
SCHEMBL3291152 0.86 BCHE (0.55) MEN1POLBMAPK1KMT2ANPSR1
SCHEMBL8935445 0.86 BCHE (0.55) MEN1POLBMAPK1KMT2ANPSR1
SCHEMBL6688641 0.85 MME (0.51) MAOBSCN9AMAOA
SCHEMBL6688644 0.85 MME (0.51) MAOBSCN9AMAOA
SCHEMBL6688332 0.84 MAOB (0.53) MAOB
SCHEMBL6688338 0.84 MAOB (0.53) MAOB
SCHEMBL6685594 0.82 SCN9A (0.50) MAOBSCN9AMAOAMEN1POLB
SCHEMBL6685589 0.82 SCN9A (0.50) MAOBSCN9AMAOAMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed