SCHEMBL6691807

SCHEMBL6691807

CS(=O)(=O)c1ccc(-c2c(-c3ccccn3)c[nH]c(=O)c2-c2ccccc2C#N)cc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.43
SCD O00767 1/20 0.41
PTGS1 P23219 2/20 0.41
TGFBR1 P36897 1/20 0.40
CBFB Q13951 1/20 0.40
GRIA1 P42261 1/20 0.39
GRIA3 P42263 1/20 0.39
PDE4D Q08499 1/20 0.39
IKBKB O14920 1/20 0.37
CHUK O15111 1/20 0.37
BRD4 O60885 1/20 0.36
GCK P35557 1/20 0.36
PTGES O14684 1/20 0.35
DYRK1B Q9Y463 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2918049 0.87 GRIA1 (0.47) GRIA1GRIA3PDE4D
Water SCHEMBL4777584 0.87 GRIA1 (0.47) GRIA1GRIA3PDE4D
SCHEMBL6686812 0.83 GRIA1 (0.47) GRIA1GRIA3PDE4D
SCHEMBL6674051 0.82 PARP1 (0.39) GRIA1GRIA3PDE4D
SCHEMBL1882884 0.80 GRIA1 (0.47) TGFBR1GRIA1GRIA3PDE4D
SCHEMBL6680176 0.79 LRRK2 (0.44) GRIA1GRIA3PDE4DIKBKBCHUK
SCHEMBL6677166 0.78 GRIA1 (0.40) GRIA1GRIA3PDE4D
SCHEMBL6689989 0.78 KDM4E (0.43) CBFBGRIA1GRIA3PDE4D
SCHEMBL6698453 0.77 GRIA1 (0.47) TGFBR1GRIA1GRIA3PDE4D
SCHEMBL2762970 0.77 MCL1 (0.50) TGFBR1GRIA1GRIA3PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465626-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES Eisai Co., Ltd. (JP) 2004-10-13 EP disclosed
WO-2003047577-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES EISAI CO LTD (JP) 2003-06-12 WO disclosed