SCHEMBL6691863

SCHEMBL6691863

CCOc1ccc(N2CCOCC2)c2sc(C(N)=O)nc12

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.52
ADORA1 P30542 16/20 0.52
ADORA2B P29275 5/20 0.48
ADORA3 P0DMS8 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2825553 0.89 ADORA2A (0.63) ADORA2AADORA1ADORA2BADORA3
SCHEMBL6691865 0.83 ADORA2A (0.46) ADORA2AADORA1ADORA2BADORA3
SCHEMBL2214868 0.79 ADORA2A (0.64) ADORA2AADORA1ADORA2BADORA3
SCHEMBL4774805 0.78 ADORA2A (0.58) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5493038 0.78 ADORA2A (0.57) ADORA2AADORA1ADORA2BADORA3
SCHEMBL20702385 0.77 ADORA2A (0.42) ADORA2AADORA1ADORA2BADORA3
SCHEMBL3052494 0.77 ADORA2A (0.48) ADORA2AADORA1ADORA2BADORA3
SCHEMBL7173118 0.76 ALDH1A1 (0.53) ADORA2AADORA1
SCHEMBL3057679 0.76 ADORA2A (0.48) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5038587 0.75 ADORA2A (0.63) ADORA2AADORA1ADORA2BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6727247-B2 ADENOSINE RECEPTOR LIGANDS IN A METHOD OF TREATMENT, CONTROL, OR PREVENTION OF CENTRAL NERVOUS SYSTEM DISORDERS HOFFMAN-LA ROCHE INC. 2004-04-27 US claimed