SCHEMBL6691865

SCHEMBL6691865

CCOc1ccc(N2CCOCC2)c2sc(N)nc12

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 17/20 0.46
ADORA1 P30542 15/20 0.46
MAPK1 P28482 2/20 0.46
KDM4E B2RXH2 1/20 0.46
HSD17B10 Q99714 1/20 0.46
PIK3CB P42338 1/20 0.43
ADORA2B P29275 4/20 0.43
ADORA3 P0DMS8 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2824784 0.86 ADORA2A (0.59) ADORA2AADORA1ADORA2BADORA3
SCHEMBL3039095 0.84 ALDH1A1 (0.46) ADORA2AADORA1MAPK1HSD17B10SMN1; SMN2
SCHEMBL6691863 0.83 ADORA2A (0.52) ADORA2AADORA1ADORA2BADORA3
SCHEMBL14217220 0.81 ADORA2A (0.41) ADORA2AADORA1ADORA2BADORA3SMN1; SMN2
SCHEMBL8358665 0.80 HPGD (0.44) ADORA2AADORA1MAPK1KDM4ESMN1; SMN2
SCHEMBL25323852 0.77 KDM4E (0.68) MAPK1KDM4EHSD17B10PIK3CBSMN1; SMN2
SCHEMBL7173118 0.74 ALDH1A1 (0.53) ADORA2AADORA1MAPK1KDM4ESMN1; SMN2
SCHEMBL14217221 0.74 MAPT (0.41) ADORA2AADORA1ADORA2BSMN1; SMN2
SCHEMBL3055076 0.74 ALDH1A1 (0.60) ADORA2AADORA1HSD17B10ADORA2BADORA3
SCHEMBL13362261 0.74 ADORA2A (0.61) ADORA2AADORA1ADORA2BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6727247-B2 ADENOSINE RECEPTOR LIGANDS IN A METHOD OF TREATMENT, CONTROL, OR PREVENTION OF CENTRAL NERVOUS SYSTEM DISORDERS HOFFMAN-LA ROCHE INC. 2004-04-27 US claimed