SCHEMBL6692478

SCHEMBL6692478

C#CCN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
KCNQ4 P56696 3/20 0.33
KCNQ5 Q9NR82 3/20 0.33
CA14 Q9ULX7 1/20 0.33
CTSD P07339 1/20 0.31
CTSL P07711 1/20 0.31
CTSB P07858 1/20 0.31
CTSS P25774 1/20 0.31
DGAT1 O75907 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22085540 0.89 CA14 (0.31) HDAC6HDAC1HDAC2KCNQ4KCNQ5
SCHEMBL1696194 0.87 HDAC6 (0.35) HDAC6HDAC1HDAC2KCNQ4KCNQ5
SCHEMBL1207293 0.83 CA14 (0.39) HDAC6HDAC1HDAC2KCNQ4KCNQ5
SCHEMBL1743767 0.82 HDAC6 (0.35) HDAC6HDAC1HDAC2KCNQ4KCNQ5
SCHEMBL10339672 0.81 HDAC6 (0.37) HDAC6HDAC1HDAC2CA14CTSD
SCHEMBL29850241 0.81 KCNQ4 (0.34) KCNQ4KCNQ5CA14
SCHEMBL15285654 0.81
SCHEMBL7073506 0.80 HDAC6 (0.34) HDAC6HDAC1HDAC2CA14DGAT1
SCHEMBL30897721 0.80 HDAC6 (0.34) HDAC6HDAC1HDAC2KCNQ4KCNQ5
SCHEMBL15286314 0.79 HDAC6 (0.32) HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025133217-A1 COMPOUNDS FLINDR THERAPEUTICS B. V. (NL) 2025-06-26 WO disclosed
US-20250188089-A1 SUBSTITUTED PYRIDOTRIAZINE COMPOUNDS AND USES THEREOF GILEAD SCIENCES, INC. 2025-06-12 US disclosed
EP-4543859-A1 3-(SULPHONYL OR SULFONIMIDOYL)PROP-2-EN-1-YL]-2-OXO-1,2-DIHYDROPYRIDINE-3-CARBOXAMIDE DERIVATIVES Flindr Therapeutics B.V. (NL) 2025-04-30 EP disclosed
US-12240828-B2 Heteroaromatic compounds as vanin inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2025-03-04 US disclosed
EP-3890828-B1 HETEROAROMATIC COMPOUNDS AS VANIN INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2025-02-19 EP disclosed
US-12187734-B2 Substituted pyridotriazine compounds and uses thereof GILEAD SCIENCES, INC. (US) 2025-01-07 US disclosed
EP-4196479-B9 SUBSTITUTED PYRIDOTRIAZINE COMPOUNDS AND USES THEREOF GILEAD SCIENCES INC (US) 2024-10-16 EP disclosed
US-20240300966-A1 SUBSTITUTED PYRIDOTRIAZINE COMPOUNDS AND USES THEREOF GILEAD SCIENCES, INC. 2024-09-12 US disclosed
EP-4321217-A2 SUBSTITUTED PYRIDOTRIAZINE COMPOUNDS AND USES THEREOF Gilead Sciences, Inc. (US) 2024-02-14 EP disclosed
US-11897892-B2 Substituted pyridotriazine compounds and uses thereof GILEAD SCIENCES, INC. (US) 2024-02-13 US disclosed
US-11613546-B2 Substituted pyridotriazine compounds and uses thereof GILEAD SCIENCES, INC. (US) 2023-03-28 US disclosed
WO-2023019166-A1 PROTEIN TYROSINE PHOSPHATASE TARGETING LIGANDS CALICO LIFE SCIENCES LLC (US) 2023-02-16 WO disclosed
WO-2023019166-A1 PROTEIN TYROSINE PHOSPHATASE TARGETING LIGANDS CALICO LIFE SCIENCES LLC (US) 2023-02-16 WO disclosed
US-20220267343-A1 SUBSTITUTED PYRIDOTRIAZINE COMPOUNDS AND USES THEREOF GILEAD SCIENCES, INC. 2022-08-25 US disclosed
WO-2022159387-A1 SUBSTITUTED PYRIDOTRIAZINE COMPOUNDS AND USES THEREOF GILEAD SCIENCES, INC. (US) 2022-07-28 WO disclosed
US-20220048889-A1 HETEROAROMATIC COMPOUNDS AS VANIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-02-17 US disclosed
US-20220048889-A1 HETEROAROMATIC COMPOUNDS AS VANIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-02-17 US disclosed
WO-2020114947-A1 HETEROAROMATIC COMPOUNDS AS VANIN INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2020-06-11 WO disclosed
US-20170174695-A1 NEW SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2017-06-22 US disclosed
WO-2004074336-A1 NOVEL CATIONIC COPOLYMERS, USE THEREOF FOR THE VECTORISATION OF BIOMOLECULES AND SYNTHETIC INTERMEDIATES FOR THE SAME HALISOL (FR) 2004-09-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12240828-B2 Heteroaromatic compounds as vanin inhibitors VHL, FANCI, PAH HDAC6 1437/4885HDAC1 1745/4885HDAC2 925/4885
US-11897892-B2 Substituted pyridotriazine compounds and uses thereof TPMT, TYMP, DPYD HDAC6 2449/4885HDAC1 1956/4885HDAC2 2542/4885
US-20170174695-A1 NEW SPIRO[3H-INDOLE-3,2'-PYRROLIDIN]-2(1H)-ONE COMPOUNDS AND DERIVATIVES AS MDM2-P53 INHIBITORS TP53, MDM2, FOXM1 HDAC6 636/4885HDAC1 394/4885HDAC2 594/4885
US-11613546-B2 Substituted pyridotriazine compounds and uses thereof TPMT, TYMP, DPYD HDAC6 2449/4885HDAC1 1956/4885HDAC2 2542/4885
US-12187734-B2 Substituted pyridotriazine compounds and uses thereof TPMT, TYMP, DPYD HDAC6 2449/4885HDAC1 1956/4885HDAC2 2542/4885
US-20250188089-A1 SUBSTITUTED PYRIDOTRIAZINE COMPOUNDS AND USES THEREOF TPMT, TYMP, DPYD HDAC6 2449/4885HDAC1 1956/4885HDAC2 2542/4885
US-20220048889-A1 HETEROAROMATIC COMPOUNDS AS VANIN INHIBITORS VHL, FANCI, PAH HDAC6 1437/4885HDAC1 1745/4885HDAC2 925/4885
US-20220267343-A1 SUBSTITUTED PYRIDOTRIAZINE COMPOUNDS AND USES THEREOF TPMT, TYMP, DPYD HDAC6 2449/4885HDAC1 1956/4885HDAC2 2542/4885
US-20240300966-A1 SUBSTITUTED PYRIDOTRIAZINE COMPOUNDS AND USES THEREOF TPMT, TYMP, DPYD HDAC6 2449/4885HDAC1 1956/4885HDAC2 2542/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.