SCHEMBL6693313

SCHEMBL6693313

CC(=O)OCC#Cc1cccc(N)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.46
IKBKB O14920 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HCRTR1 O43613 1/20 0.36
ALOX5 P09917 1/20 0.36
ASIC3 Q9UHC3 1/20 0.36
ADRB2 P07550 3/20 0.36
ADRB1 P08588 2/20 0.36
ADRB3 P13945 2/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
PTPRC P08575 1/20 0.36
PTPRG P23470 1/20 0.36
RAB9A P51151 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CSNK2A2 P19784 1/20 0.35
CSNK2B P67870 1/20 0.35
CSNK2A1 P68400 1/20 0.35
MMP1 P03956 1/20 0.35
MMP2 P08253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6689174 0.83 FFAR1 (0.42) FFAR1ALDH1A1ASIC3DRD2DRD3
SCHEMBL27545848 0.80 ALDH1A1 (0.48) FFAR1ALDH1A1MMP2MMP12
SCHEMBL6696133 0.77 ALDH1A1 (0.51) FFAR1ALDH1A1
SCHEMBL13529219 0.76 CYP3A4 (0.43) FFAR1ALDH1A1HCRTR1ASIC3ADRB2
SCHEMBL2150674 0.74 FFAR1 (0.50) FFAR1IKBKBALDH1A1HCRTR1ALOX5
SCHEMBL2810465 0.73 FFAR1 (0.44) FFAR1IKBKBALDH1A1HCRTR1ASIC3
SCHEMBL13529220 0.73 FFAR1 (0.47) FFAR1IKBKBALDH1A1HCRTR1ASIC3
SCHEMBL6694265 0.72 FFAR1 (0.62) FFAR1IKBKBASIC3DRD2DRD3
Ethyl Acetate SCHEMBL27988644 0.72 ALDH1A1 (0.54) ALDH1A1RAB9AL3MBTL1
SCHEMBL75802 0.71 CYP2D6 (0.45) ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004106292-A1 HALOETHYL UREA COMPOUNDS AND THEIR USE TO ATTENUATE, INHIBIT OR PREVENT NON-CANCEROUS PATHOGENIC CELLULAR PROLIFERATION AND DISEASES ASSOCIATED THEREWITH IMOTEP INC. (CA) 2004-12-09 WO disclosed
WO-2004106291-A1 HALOETHYL UREA COMPOUNDS AND THE USE THEREOF TO ATTENUATE, INHIBIT OR PREVENT CANCER CELL MIGRATION IMOTEP INC. (CA) 2004-12-09 WO disclosed