SCHEMBL6693458

SCHEMBL6693458

COc1ccc(-n2nc(OC3CCCC3)nc2-c2ccc(Br)cc2)cn1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.42
PTGS2 P35354 4/20 0.42
PDE4D Q08499 1/20 0.40
MALT1 Q9UDY8 1/20 0.39
OXTR P30559 10/20 0.37
AVPR1A P37288 8/20 0.37
AVPR2 P30518 2/20 0.36
CHRNB2 P17787 3/20 0.34
CHRNA4 P43681 3/20 0.34
CHRNB4 P30926 2/20 0.34
CHRNA3 P32297 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6682055 0.90 PTGS1 (0.42) PTGS1PTGS2OXTRAVPR1AAVPR2
SCHEMBL6687338 0.90 PTGS1 (0.42) PTGS1PTGS2PDE4DOXTRAVPR1A
SCHEMBL6682526 0.87 PTGS1 (0.40) PTGS1PTGS2OXTRAVPR1AAVPR2
SCHEMBL6682120 0.87 PTGS1 (0.40) PTGS1PTGS2OXTRAVPR1AAVPR2
SCHEMBL6682517 0.83 PTGS1 (0.41) PTGS1PTGS2OXTRAVPR1AAVPR2
SCHEMBL6687070 0.81 GRIA2 (0.36) PTGS1PTGS2MALT1OXTRAVPR1A
SCHEMBL6682093 0.80 MALT1 (0.41) PTGS1PTGS2PDE4DMALT1MEN1
SCHEMBL6132456 0.78 PTGS2 (0.67) PTGS1PTGS2PDE4DMALT1
SCHEMBL6681645 0.78 PTGS1 (0.40) PTGS1PTGS2MALT1OXTRAVPR1A
SCHEMBL6681046 0.73 PTGS2 (0.60) PTGS1PTGS2PDE4DMALT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004060367-A1 IMIDAZOLE AND TRIAZOLE DERIVATIVES USEFUL AS SELECTIVE COX-1 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-07-22 WO disclosed