SCHEMBL6681645

SCHEMBL6681645

COc1ccc(-n2nc(O)nc2-c2ccc(Br)cc2)cn1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.40
PTGS2 P35354 4/20 0.40
MALT1 Q9UDY8 1/20 0.39
OXTR P30559 3/20 0.39
AVPR2 P30518 2/20 0.39
AVPR1A P37288 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP2A6 P11509 1/20 0.37
HSD17B1 P14061 1/20 0.36
HSD17B2 P37059 1/20 0.36
MAPT P10636 1/20 0.36
JAK2 O60674 1/20 0.36
FYN P06241 1/20 0.36
GPR183 P32249 1/20 0.35
ACLY P53396 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6132556 0.89 PTGS2 (0.53) PTGS1PTGS2MALT1OXTRAVPR2
SCHEMBL6135189 0.81 PTGS2 (0.53) PTGS1PTGS2MALT1OXTRCYP2A6
SCHEMBL6687139 0.80 MEN1 (0.48) PTGS1PTGS2OXTRAVPR2AVPR1A
SCHEMBL6693458 0.78 PTGS1 (0.42) PTGS1PTGS2MALT1OXTRAVPR2
SCHEMBL6680327 0.76 PTGS1 (0.45) PTGS1PTGS2OXTRAVPR2AVPR1A
SCHEMBL6686662 0.75 PTGS1 (0.47) PTGS1PTGS2MALT1OXTRAVPR2
SCHEMBL4028727 0.74 PTGS2 (0.69) PTGS1PTGS2MALT1
SCHEMBL5782756 0.73 SMN1; SMN2 (0.51) PTGS2MALT1MEN1KMT2AMAPT
SCHEMBL5781861 0.72 L3MBTL1 (0.44) PTGS2MALT1MEN1KMT2AMAPT
SCHEMBL6687276 0.72 L3MBTL1 (0.42) PTGS1PTGS2MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004060367-A1 IMIDAZOLE AND TRIAZOLE DERIVATIVES USEFUL AS SELECTIVE COX-1 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-07-22 WO disclosed