SCHEMBL669491

SCHEMBL669491

CC(C)(C)OC(=O)NC(=O)N1CCCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.45
HPGD P15428 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
ALOX15 P16050 1/20 0.41
HTT P42858 1/20 0.41
MAPT P10636 1/20 0.40
GAA P10253 2/20 0.39
PREP P48147 1/20 0.39
EPHX2 P34913 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
USP2 O75604 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3880063 0.98 CTSK (0.46) CTSKHPGDCA1CA2SMN1; SMN2
SCHEMBL945981 0.96 MAPT (0.43) CTSKHPGDCA1CA2SMN1; SMN2
SCHEMBL4738498 0.84 EPHX2 (0.38) CTSKHPGDCA1CA2SMN1; SMN2
SCHEMBL7040760 0.76 CTSK (0.38) CTSKHPGDCA1CA2SMN1; SMN2
SCHEMBL7040763 0.76 CTSK (0.38) CTSKHPGDCA1CA2SMN1; SMN2
SCHEMBL8191259 0.75 HPGD (0.39) CTSKHPGDCA1CA2GAA
SCHEMBL8191256 0.75 HPGD (0.39) CTSKHPGDCA1CA2GAA
SCHEMBL2025016 0.74 HPGD (0.47) CTSKHPGDCA1CA2SMN1; SMN2
SCHEMBL9106442 0.74 HPGD (0.41) CTSKHPGDCA1CA2SMN1; SMN2
Ethyne SCHEMBL9752605 0.74 HPGD (0.64) CTSKHPGDSMN1; SMN2MAPTPREP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2606038-B1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2016-01-13 EP claimed
US-8765944-B2 Compounds for the treatment of hepatitis C BRISTOL-MYERS SQUIBB COMPANY (US) 2014-07-01 US claimed
EP-2606038-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-06-26 EP claimed
US-20120213729-A1 Compounds for the Treatment of Hepatitis C BRISTOL-MYERS SQUIBB COMPANY 2012-08-23 US claimed
WO-2012024373-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2012-02-23 WO claimed
WO-2024137742-A1 COMPOUNDS AND COMPOSITIONS AS FGFR3 DEGRADERS AND USES THEREOF BLUEPRINT MEDICINES CORPORATION (US) 2024-06-27 WO disclosed
EP-2606038-B1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2016-01-13 EP disclosed
US-8765944-B2 Compounds for the treatment of hepatitis C BRISTOL-MYERS SQUIBB COMPANY (US) 2014-07-01 US disclosed
EP-2606038-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-06-26 EP disclosed
US-20120213729-A1 Compounds for the Treatment of Hepatitis C BRISTOL-MYERS SQUIBB COMPANY 2012-08-23 US disclosed
WO-2012024373-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2012-02-23 WO disclosed
EP-1380582-B1 FSH mimetics for the treatment of infertility APPLIED RESEARCH SYSTEMS (AN) 2006-06-14 EP disclosed
EP-1102763-B1 FSH MIMETICS FOR THE TREATMENT OF INFERTILITY APPLIED RESEARCH SYSTEMS (AN) 2004-10-13 EP disclosed
EP-1380582-A1 FSH mimetics for the treatment of infertility Applied Research Systems ARS Holding N.V. (AN) 2004-01-14 EP disclosed
US-6653338-B2 Heterocyclic carboxamide compounds APPLIED RESEARCH SYSTEMS ARS HOLDING N.A. (NL) 2003-11-25 US disclosed
US-20020147345-A1 FSH mimetics for the treatment of infertility MERCK SERONO SA (CH) 2002-10-10 US disclosed
US-6423723-B1 ORAL BIOAVAILABILITY APPLIED RESEARCH SYSTEMS ARS HOLDING N. A. (NL) 2002-07-23 US disclosed
EP-1102763-A2 FSH MIMETICS FOR THE TREATMENT OF INFERTILITY Applied Research Systems ARS Holding N.V. (AN) 2001-05-30 EP disclosed
US-6235755-B1 FOLLICLE STIMULATING HORMONE ANTAGONIST APPLIED RESEARCH SYSTEMS ARS HOLDING N.A. (AN) 2001-05-22 US disclosed
WO-2000008015-A2 FSH MIMETICS FOR THE TREATMENT OF INFERTILITY APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2000-02-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020147345-A1 FSH mimetics for the treatment of infertility FSHR, GNRHR, LHCGR CTSK 2023/4885HPGD 3083/4885CA1 3182/4885
US-20120213729-A1 Compounds for the Treatment of Hepatitis C HAVCR2, SLC10A1, HCCS CTSK 520/4885HPGD 1433/4885CA1 4446/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.