SCHEMBL6694933

SCHEMBL6694933

NC=CCc1cccc2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.48
CYP2C19 P33261 3/20 0.48
CYP2C9 P11712 1/20 0.48
HPGD P15428 3/20 0.47
HTT P42858 2/20 0.47
CYP2D6 P10635 3/20 0.46
TDP1 Q9NUW8 1/20 0.44
CA2 P00918 1/20 0.43
ACP3 P15309 1/20 0.43
MTNR1A P48039 1/20 0.41
TSHR P16473 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NR1I2 O75469 1/20 0.41
DRD2 P14416 1/20 0.41
ADRA2C P18825 1/20 0.41
CNR1 P21554 1/20 0.41
SLC6A2 P23975 1/20 0.41
HTR2A P28223 1/20 0.41
SLC6A4 P31645 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2136855 0.84 CYP2C19 (0.50) CYP1A2CYP2C19CYP2C9HPGDHTT
SCHEMBL1611481 0.84 CYP2C19 (0.50) CYP1A2CYP2C19CYP2C9HPGDHTT
SCHEMBL7648676 0.83 CYP2C19 (0.52) CYP1A2CYP2C19CYP2C9HPGDHTT
SCHEMBL666674 0.80 MAOB (0.38) HTR2A
SCHEMBL10499434 0.80 CYP1A2 (0.48) CYP1A2CYP2C19CYP2C9HPGDHTT
SCHEMBL7924285 0.80 CYP2C19 (0.48) CYP1A2CYP2C19CYP2C9HPGDHTT
SCHEMBL301409 0.80 CYP2C19 (0.48) CYP1A2CYP2C19CYP2C9HPGDHTT
SCHEMBL4229398 0.80 CYP2C19 (0.48) CYP1A2CYP2C19CYP2C9HPGDHTT
SCHEMBL1325661 0.80 TDP1 (0.48) CYP1A2CYP2C19CYP2C9HPGDHTT
SCHEMBL3801024 0.79 ALDH1A1 (0.41) CYP1A2CYP2C19CYP2C9HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105925124-A Anticorrosive Coating Composition, Anticorrosive Coating Film, Substrate With Anticorrosive Coating Film, And Method For Producing Substrate With Anticorrosive Coating Film 中国涂料株式会社 2016-09-07 CN disclosed
CN-101001929-A High-solid anticorrosive coating composition, high-solid rapidly-curable anticorrosive coating composition, method of coating ship or the like, high-solid anticorrosive film and rapidly cured high-sol CHUGOKU MARINE PAINTS (JP) 2007-07-18 CN disclosed
EP-1027043-B1 BENZODIOXOLE, BENZOFURAN, DIHYDROBENZOFURAN, AND BENZODIOXANE MELATONERGIC AGENTS BRISTOL MYERS SQUIBB CO (US) 2004-11-10 EP disclosed
EP-1027043-A4 BENZODIOXOLE, BENZOFURAN, DIHYDROBENZOFURAN, AND BENZODIOXANE MELATONERGIC AGENTS BRISTOL MYERS SQUIBB CO (US) 2002-02-20 EP disclosed
EP-1027043-A1 BENZODIOXOLE, BENZOFURAN, DIHYDROBENZOFURAN, AND BENZODIOXANE MELATONERGIC AGENTS Bristol-Myers Squibb Company (US) 2000-08-16 EP disclosed
US-6028112-A Spirocyclopropyl fluorenes as melatonergic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-02-22 US disclosed
US-5981571-A USEFUL AS MELATONERGIC AGENTS IN THE TREATMENT OF SLEEP DISORDERS, SEASONAL DEPRESSION, SHIFTS IN CIRCADIAN CYCLES, MELANCHOLIA, STRESS, APPETITE REGULATION, BENIGN PROSTATIC HYPERPLASIA AND RELATED CONDITIONS BRISTOL-MYERS SQUIBB COMPANY (US) 1999-11-09 US disclosed
US-5856529-A ADJUSTMENT OF NERVOUS SYSTEM, ENDOCRINE FUNCTION; REPRODUCTION, BODY WEIGHT AND METABOLISM BRISTOL-MYERS SQUIBB COMPANY (US) 1999-01-05 US disclosed
WO-1998052554-A1 SPIROCYCLOPROPYL FLUORENES AS MELATONERGIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-11-26 WO disclosed
EP-0718286-B1 3-Alkoxybenzylpiperidine derivatives as melatonergic agents BRISTOL MYERS SQUIBB CO (US) 1998-07-29 EP disclosed
US-5661185-A AN ALKOXYPHENYL-ALKYLUREA COMPOUND TREATING SLEEP DISORDER BRISTOL-MYERS SQUIBB CO. (US) 1997-08-26 US disclosed
EP-0728738-A1 Tetralinyl- and indanyl-ethylamides having melatonergic activity BRISTOL-MYERS SQUIBB COMPANY (US) 1996-08-28 EP disclosed
US-5541228-A Melatonergic agents BRISTOL-MYERS SQUIBB CO. (US) 1996-07-30 US disclosed
EP-0718286-A1 3-Alkoxybenzylpiperidine derivatives as melatonergic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1996-06-26 EP disclosed
US-5530012-A FOR SLEEP DISORDERS, DEPRESSION, GLAUCOMA, CANCER BRISTOL-MYERS SQUIBB CO. (US) 1996-06-25 US disclosed
EP-0706994-A1 Melatonergic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1996-04-17 EP disclosed
US-5318994-A Treating melatoninergic disorders ADIR ET COMPAGNIE (FR) 1994-06-07 US disclosed
US-5225442-A Melatoninergic disorders ADIR ET COMPAGNIE (FR) 1993-07-06 US disclosed
US-5194614-A COMPOUNDS HAVING A NAPHTHALENE STRUCTURE ADIR ET COMPAGNIE (FR) 1993-03-16 US disclosed
EP-0100257-A2 Aminoalkyl naphthalene derivatives, their salts, process for their preparation and the therapeutical use of these derivatives and salts DELALANDE S.A. (FR) 1984-02-08 EP disclosed