SCHEMBL6701211

SCHEMBL6701211

CCOC(=O)CN1CCN(c2ccc(C(N)=O)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.53
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
HTT P42858 2/20 0.53
CHRNA7 P36544 1/20 0.52
CHRNA10 Q9GZZ6 1/20 0.52
CHRNA9 Q9UGM1 1/20 0.52
TSHR P16473 2/20 0.50
SMN1; SMN2 Q16637 4/20 0.49
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48
POLB P06746 2/20 0.48
MAPT P10636 6/20 0.48
LMNA P02545 4/20 0.48
KDM4E B2RXH2 1/20 0.48
GAA P10253 1/20 0.48
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7356492 0.86 F2 (0.52) ALDH1A1TSHRSMN1; SMN2ITGB3ITGA2B
SCHEMBL6701215 0.86 MAPT (0.58) ALDH1A1MEN1KMT2ATSHRSMN1; SMN2
SCHEMBL20271748 0.83 ALDH1A1 (0.56) ALDH1A1MEN1KMT2AHTTSMN1; SMN2
SCHEMBL20271984 0.83 SMN1; SMN2 (0.69) ALDH1A1MEN1KMT2AHTTTSHR
SCHEMBL14860445 0.83 ALDH1A1 (0.60) ALDH1A1MEN1KMT2AHTTCHRNA7
SCHEMBL31050602 0.82 ALDH1A1 (0.53) ALDH1A1MEN1KMT2ATSHRSMN1; SMN2
SCHEMBL27456657 0.82 MAPT (0.71) ALDH1A1MEN1KMT2AHTTCHRNA7
SCHEMBL2232683 0.81 GAA (0.62) ALDH1A1MEN1KMT2AHTTCHRNA7
SCHEMBL6698448 0.81 ALDH1A1 (0.61) ALDH1A1MEN1KMT2AHTTCHRNA7
SCHEMBL20271985 0.80 PPARD (0.51) ALDH1A1SMN1; SMN2MAPTLMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1135378-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS APOB-100 SECRETION INHIBITORS GLAXO GROUP LIMITED (GB) 2001-09-26 EP claimed
WO-2000032582-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS APOB-100 SECRETION INHIBITORS GLAXO GROUP LIMITED (GB) 2000-06-08 WO claimed
US-20040044008-A1 Use of therapeutic benzamide derivatives DAUGAN ALAIN CLAUDE-MARIE (FR) 2004-03-04 US disclosed
WO-2003048121-A1 THERAPEUTIC BENZAMIDE DERIVATIVES GLAXO GROUP LIMITED (GB) 2003-06-12 WO disclosed
US-6552022-B1 Atherosclerosis in a mammal, pancreatitis, non-insulin dependent diabetes mellitus, coronary heart disease in a lowering serum lipid levels SMITHKLINE BEECHAM CORPORATION 2003-04-22 US disclosed
EP-1286670-A2 USE OF THERAPEUTIC BENZAMIDE DERIVATIVES GLAXO GROUP LIMITED (GB) 2003-03-05 EP disclosed
WO-2001097810-A2 USE OF THERAPEUTIC BENZAMIDE DERIVATIVES GLAXO GROUP LIMITED (GB) 2001-12-27 WO disclosed
EP-1135378-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS APOB-100 SECRETION INHIBITORS GLAXO GROUP LIMITED (GB) 2001-09-26 EP disclosed
WO-2000032582-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS APOB-100 SECRETION INHIBITORS GLAXO GROUP LIMITED (GB) 2000-06-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040044008-A1 Use of therapeutic benzamide derivatives MTTP, LIPC, CETP ALDH1A1 379/4885MEN1 3940/4885KMT2A 1929/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.