Cyclohexanone

Cyclohexanone

SCHEMBL670911

CS(=O)(=O)O.O=C1CCCCC1

nearest known ligand 0.61

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Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of Cyclohexanone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRIM24 O15164 2/20 0.61
TRIM33 Q9UPN9 2/20 0.61
ALDH1A1 P00352 2/20 0.61
SLC2A1 P11166 1/20 0.34
KMT2A Q03164 1/20 0.32
CA2 P00918 1/20 0.32
ALOX15 P16050 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cyclooctanone SCHEMBL28121636 0.88 TRIM24 (0.69) TRIM24TRIM33ALDH1A1
Cyclohexanone SCHEMBL29032564 0.88 TRIM24 (0.69) TRIM24TRIM33ALDH1A1
Cyclohexanone SCHEMBL28691080 0.86 TRIM24 (0.65) TRIM24TRIM33ALDH1A1
Methyl Alcohol SCHEMBL5716663 0.82 TRIM24 (0.79) TRIM24TRIM33ALDH1A1KMT2ACA2
Cyclohexanone SCHEMBL16238114 0.82 TRIM24 (0.79) TRIM24TRIM33ALDH1A1KMT2ACA2
Cyclohexanone SCHEMBL1961575 0.82
Cyclohexanone SCHEMBL28313315 0.81 TRIM24 (0.58) TRIM24TRIM33ALDH1A1
Cyclohexanone SCHEMBL27541062 0.79 TRIM24 (0.73) TRIM24TRIM33ALDH1A1KMT2ACA2
Cyclohexanone SCHEMBL10924657 0.79 TRIM24 (0.73) TRIM24TRIM33ALDH1A1KMT2ACA2
Cyclopentanone SCHEMBL21611329 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2605772-B1 PROCESS FOR PREPARING AMINOCYCLOHEXYL ETHER COMPOUNDS CARDIOME INTERNAT AG (CH) 2016-06-22 EP disclosed
US-20150259284-A1 PROCESS FOR PREPARING AMINOCYCLOHEXYL ETHER COMPOUNDS CARDIOME INTERNATIONAL SA (CH) 2015-09-17 US disclosed
US-9006460-B2 Process for preparing aminocyclohexyl ether compounds CARDIOME INTERNATIONAL AG (CH) 2015-04-14 US disclosed
EP-2605772-A2 PROCESS FOR PREPARING AMINOCYCLOHEXYL ETHER COMPOUNDS Merck Sharp & Dohme Corp. (US) 2013-06-26 EP disclosed
US-20130149751-A1 PROCESS FOR PREPARING AMINOCYCLOHEXYL ETHER COMPOUNDS CARDIOME INTERNATIONAL SA (CH) 2013-06-13 US disclosed
WO-2012024100-A2 PROCESS FOR PREPARING AMINOCYCLOHEXYL ETHER COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2012-02-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150259284-A1 PROCESS FOR PREPARING AMINOCYCLOHEXYL ETHER COMPOUNDS CYP3A43, CYP4B1, CYP3A4 TRIM24 2772/4885TRIM33 2483/4885ALDH1A1 393/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.