SCHEMBL6712438

SCHEMBL6712438

Cc1ccc(S(=O)(=O)NC(=O)c2cc(C)c3nc(C)n(Cc4ccc(N5CCCCCC5)cc4Cl)c3n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.39
ALDH1A1 P00352 3/20 0.39
TP53 P04637 2/20 0.39
KDM4E B2RXH2 2/20 0.39
GLA P06280 1/20 0.39
CYP3A4 P08684 1/20 0.39
GAA P10253 1/20 0.39
ALOX12 P18054 1/20 0.39
NFKB1 P19838 1/20 0.39
RECQL P46063 1/20 0.38
EPHX2 P34913 3/20 0.38
NR1H4 Q96RI1 3/20 0.38
PTGS2 P35354 2/20 0.38
PTGS1 P23219 1/20 0.38
TRPV1 Q8NER1 2/20 0.37
FLT1 P17948 1/20 0.36
FLT4 P35916 1/20 0.36
KDR P35968 1/20 0.36
KMT2A Q03164 1/20 0.35
EGFR P00533 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6306260 1.00 MAPT (0.39) MAPTALDH1A1TP53KDM4EGLA
SCHEMBL6306800 0.99 PTGS2 (0.38) MAPTALDH1A1TP53KDM4EGLA
SCHEMBL6305528 0.93 PTGS2 (0.37) ALDH1A1TP53KDM4EPTGS2PTGS1
SCHEMBL6134585 0.92 PIK3CB (0.42) MAPTALDH1A1KDM4EEPHX2NR1H4
SCHEMBL6298633 0.85 FLT1 (0.42) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL6299197 0.85 FLT1 (0.41) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL6493067 0.85 PTGS2 (0.41) MAPTALDH1A1RECQLPTGS2PTGS1
SCHEMBL6135088 0.85 PTGS2 (0.41) PTGS2PTGS1FLT1FLT4KDR
SCHEMBL6299750 0.84 PTGS2 (0.40) MAPTALDH1A1TP53PTGS2PTGS1
SCHEMBL6299098 0.83 PPARG (0.44) MAPTPTGS2PTGS1FLT1FLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040180947-A1 hypoglycemic activity or phoshodiesterase-V inhibitory activity; prophylaxis and treatment of impaired glucose tolerance disorder, diabetes (e.g., type II diabetes), diabetic complications FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-09-16 US disclosed
US-6348474-B1 COMPOUNDS AS ANTIDIABETIC AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-02-19 US disclosed
EP-0995742-A1 SULFONAMIDE COMPOUNDS AND MEDICINAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040180947-A1 hypoglycemic activity or phoshodiesterase-V inhibitory activity; prophylaxis and treatment of impaired glucose tolerance disorder, diabetes (e.g., type II diabetes), diabetic complications PDE2A, PDE3A, PYGM MAPT 4725/4885ALDH1A1 1067/4885TP53 4849/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.