SCHEMBL6714477

SCHEMBL6714477

C=CCC(N)c1cc(F)ccc1-c1noc2cc(Cl)ccc12

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.33
ESR2 Q92731 6/20 0.33
HSP90AA1 P07900 2/20 0.33
PDCD1LG2 Q9BQ51 2/20 0.31
CD274 Q9NZQ7 2/20 0.31
ALDH1A1 P00352 2/20 0.31
DPP4 P27487 1/20 0.31
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6712688 0.85 ESR1 (0.38) ESR1ESR2HSP90AA1PDCD1LG2CD274
SCHEMBL6710249 0.85 ESR1 (0.42) ESR1ESR2HSP90AA1PDCD1LG2CD274
SCHEMBL6713956 0.85 ESR1 (0.42) ESR1ESR2HSP90AA1PDCD1LG2CD274
SCHEMBL6714537 0.85 ESR1 (0.42) ESR1ESR2HSP90AA1PDCD1LG2CD274
SCHEMBL6712687 0.85 ESR1 (0.38) ESR1ESR2HSP90AA1PDCD1LG2CD274
SCHEMBL7559972 0.85 ESR1 (0.37) ESR1ESR2HSP90AA1
Hydrochloric Acid SCHEMBL2474476 0.84 ESR1 (0.37) ESR1ESR2HSP90AA1PDCD1LG2CD274
Hydrochloric Acid SCHEMBL2474474 0.84 ESR1 (0.37) ESR1ESR2HSP90AA1PDCD1LG2CD274
Hydrochloric Acid SCHEMBL6712745 0.84 ESR1 (0.37) ESR1ESR2HSP90AA1PDCD1LG2CD274
SCHEMBL6709980 0.83 ESR1 (0.38) ESR1ESR2HSP90AA1PDCD1LG2CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040229910-A1 Therapeutic compounds N.V. ORGANON (NL) 2004-11-18 US disclosed
EP-0898566-B1 SUBSTITUTED BENZYLAMINES AND THEIR USE FOR THE TREATMENT OF DEPRESSION AKZO NOBEL NV (NL) 2002-11-06 EP disclosed
US-20020037885-A1 Therapeutic compounds DIJCKS FREDERICUS ANTONIUS (NL) 2002-03-28 US disclosed
US-6313139-B1 ADMINISTERING BENZYLAMINE DERIVATIVE FOR THERAPY OF PSYCHIATRIC DISORDER IN MAMMALS AKZO NOBEL N. V. (NL) 2001-11-06 US disclosed
US-6080773-A USEFUL FOR TREATMENT OF DEPRESSION, ANXIETY OR PSYCHOSIS AKZO NOBEL, N.V. (NL) 2000-06-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040229910-A1 Therapeutic compounds BDNF, PNMT, SLC18A2 ESR1 2865/4885ESR2 1589/4885HSP90AA1 2140/4885
US-20020037885-A1 Therapeutic compounds BDNF, PNMT, SLC18A2 ESR1 2865/4885ESR2 1589/4885HSP90AA1 2140/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.