SCHEMBL6718330

SCHEMBL6718330

CC(C)(C)OC(=O)Nc1ccc(CN(Cc2ccc(C(F)(F)F)cc2)C(=O)C(=O)O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 1/20 0.49
CYP17A1 P05093 1/20 0.48
P2RY14 Q15391 1/20 0.43
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
EPHX2 P34913 1/20 0.41
UTS2R Q9UKP6 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
MMP1 P03956 1/20 0.41
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
MMP8 P22894 1/20 0.41
MMP13 P45452 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
MEN1 O00255 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4326881 0.88 CTSL (0.51) CYP17A1ALDH1A1PTGDR2MMP1MMP2
SCHEMBL1854425 0.87 NPSR1 (0.46) MTORCYP17A1PPARGPPARAALDH1A1
SCHEMBL1853151 0.83 CYP17A1 (0.54) MTORCYP17A1PPARGPPARAMAPT
SCHEMBL1854428 0.82 MTOR (0.42) MTORCYP17A1P2RY14PPARGPPARA
SCHEMBL1138925 0.82 EPHX2 (0.59) CYP17A1P2RY14ALDH1A1MAPTLMNA
SCHEMBL1854866 0.76 KCNQ3 (0.54) MTORALDH1A1MAPTSMN1; SMN2
SCHEMBL1851161 0.76 CTSL (0.49) CYP17A1PPARGPPARAALDH1A1PTGDR2
SCHEMBL30929531 0.76 EPHX2 (0.51) CYP17A1P2RY14MAPTLMNAHTT
SCHEMBL22930812 0.76 CYP17A1 (0.57) CYP17A1PPARGPPARAPTGDR2MMP1
SCHEMBL1854194 0.75 PLK1 (0.58) TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1470102-A1 SUBSTITUTED METHYLENE AMIDE DERIVATIVES AS MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPS) Applied Research Systems ARS Holding N.V. (AN) 2004-10-27 EP disclosed
WO-2003064376-A1 SUBSTITUTED METHYLENE AMIDE DERIVATIVES AS MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPS) APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2003-08-07 WO disclosed