SCHEMBL6720377

SCHEMBL6720377

O=C(O)c1c(O)c2cc(C(O)c3ccc(F)cc3)ccc2oc1=O

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 3/20 0.45
CA12 O43570 3/20 0.43
CA9 Q16790 3/20 0.43
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
GPR35 Q9HC97 1/20 0.38
TOP2A P11388 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 1/20 0.35
MGAM O43451 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6720374 0.83 CA12 (0.43) NQO1CA12CA9NPC1RAB9A
SCHEMBL6720338 0.80 NQO1 (0.53) NQO1CA12CA9NPC1RAB9A
SCHEMBL6720354 0.71 NQO1 (0.43) NQO1CA12CA9NPC1RAB9A
SCHEMBL6720336 0.69 NQO1 (0.64) NQO1CA12CA9NPC1RAB9A
SCHEMBL24864998 0.69 NQO1 (0.57) NQO1CA12CA9NPC1RAB9A
SCHEMBL29901650 0.69 CA12 (0.73) NQO1CA12CA9GPR35LMNA
SCHEMBL1648027 0.69 CA12 (0.73) NQO1CA12CA9GPR35LMNA
SCHEMBL31604852 0.69 SLC26A4 (0.51) NPC1RAB9ALMNAHTTMEN1
SCHEMBL6720324 0.69 NQO1 (0.52) NQO1CA12CA9GPR35LMNA
SCHEMBL13284846 0.68 CYP2C9 (0.65) NQO1MEN1KMT2AALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8183236-B2 Compounds with HIV-1 integrase inhibitory activity and use thereof as anti-HIV/AIDS therapeutics UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2012-05-22 US disclosed
US-8183236-B2 Compounds with HIV-1 integrase inhibitory activity and use thereof as anti-HIV/AIDS therapeutics UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2012-05-22 US disclosed
US-20090088420-A1 COMPOUNDS WITH HIV-1 INTEGRASE INHIBITORY ACTIVITY AND USE THEREOF AS ANTI-HIV/AIDS THERAPEUTICS UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2009-04-02 US disclosed
US-20090088420-A1 COMPOUNDS WITH HIV-1 INTEGRASE INHIBITORY ACTIVITY AND USE THEREOF AS ANTI-HIV/AIDS THERAPEUTICS UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2009-04-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090088420-A1 COMPOUNDS WITH HIV-1 INTEGRASE INHIBITORY ACTIVITY AND USE THEREOF AS ANTI-HIV/AIDS THERAPEUTICS TYMP, IMPDH1, SAMHD1 NQO1 437/4885CA12 4839/4885CA9 4070/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.