SCHEMBL6725294

SCHEMBL6725294

CCCCCCCCCCCc1nc(-c2ccc(CNCc3ccc(C(F)(F)F)cc3)cc2)no1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.62
S1PR3 Q99500 2/20 0.62
S1PR2 O95136 1/20 0.62
LPAR2 Q9HBW0 1/20 0.62
HDAC1 Q13547 6/20 0.61
HDAC8 Q9BY41 4/20 0.61
SIRT2 Q8IXJ6 1/20 0.60
HDAC2 Q92769 4/20 0.59
SPHK1 Q9NYA1 5/20 0.51
PPARA Q07869 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1856614 0.99 S1PR1 (0.61) S1PR1S1PR3S1PR2LPAR2HDAC1
SCHEMBL15705335 0.85 S1PR2 (0.78) S1PR1S1PR3S1PR2LPAR2HDAC1
SCHEMBL5047433 0.85 SIRT2 (0.58) S1PR1S1PR3S1PR2LPAR2HDAC1
SCHEMBL1855651 0.82 HDAC1 (0.43) S1PR1S1PR3S1PR2LPAR2HDAC1
SCHEMBL1853070 0.82 HDAC1 (0.43) S1PR1S1PR3S1PR2LPAR2HDAC1
SCHEMBL1853227 0.82 HDAC8 (0.64) S1PR1S1PR3S1PR2LPAR2HDAC1
SCHEMBL1851267 0.82 HDAC8 (0.58) S1PR1S1PR3S1PR2LPAR2HDAC1
SCHEMBL1855183 0.80 SPHK1 (0.51) S1PR1S1PR3S1PR2LPAR2HDAC1
SCHEMBL6725380 0.80 SPHK1 (0.51) S1PR1S1PR3S1PR2LPAR2HDAC1
SCHEMBL5047430 0.80 HDAC8 (0.53) S1PR1S1PR3S1PR2LPAR2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1470102-A1 SUBSTITUTED METHYLENE AMIDE DERIVATIVES AS MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPS) Applied Research Systems ARS Holding N.V. (AN) 2004-10-27 EP disclosed
WO-2003064376-A1 SUBSTITUTED METHYLENE AMIDE DERIVATIVES AS MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPS) APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2003-08-07 WO disclosed