SCHEMBL6740873

SCHEMBL6740873

CCCn1ncc2ccc(CCOS(C)(=O)=O)cc21

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMO O15229 5/20 0.39
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
HTR2B P41595 2/20 0.36
PDE1A P54750 2/20 0.36
PDE1B Q01064 2/20 0.36
PDE1C Q14123 2/20 0.36
QPCT Q16769 1/20 0.36
PLA2G4A P47712 1/20 0.36
MCHR1 Q99705 1/20 0.34
SLC16A3 O15427 2/20 0.33
SLC16A1 P53985 2/20 0.33
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.33
RAB9A P51151 1/20 0.33
BRD4 O60885 3/20 0.33
CACNA1H O95180 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19159359 0.81 HTR2A (0.45) KMOHTR2AHTR2CHTR2BPDE1A
SCHEMBL6740869 0.79 KMO (0.38) KMOHTR2AHTR2CHTR2BPDE1A
SCHEMBL31638076 0.78 CTNNB1 (0.51) HTR2APDE1CCACNA1H
SCHEMBL5792520 0.76 KMO (0.40) KMOHTR2AHTR2CHTR2BPLA2G4A
SCHEMBL27165385 0.76 HTR2A (0.51) KMOHTR2AHTR2CHTR2BQPCT
SCHEMBL27165379 0.75 HTR2A (0.54) KMOHTR2AHTR2CHTR2BMCHR1
SCHEMBL17504300 0.75 KMO (0.55) KMOHTR2AHTR2CHTR2BQPCT
SCHEMBL6746000 0.74 HRH3 (0.40) KMOHTR2AHTR2CHTR2BPDE1A
SCHEMBL6741339 0.73 HRH3 (0.50) MCHR1POLB
SCHEMBL6744654 0.73 QPCT (0.38) KMOHTR2AHTR2CHTR2BQPCT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040167158-A1 Heterocyclic compounds for the treatment of migraine NPS ALLELIX BIOPHARMACEUTICALS, INC. (CA) 2004-08-26 US disclosed
US-6716837-B1 INDOLE AND INDAZOLE COMPOUNDS NPS ALLELIX BIOPHARMACEUTICALS, INC. (CA) 2004-04-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040167158-A1 Heterocyclic compounds for the treatment of migraine SCN7A, CNR2, HTR7 KMO 453/4885HTR2A 294/4885HTR2C 116/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.