SCHEMBL6741465

SCHEMBL6741465

[CH2]c1cc(C)cc(C#N)c1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
CYP2A6 P11509 1/20 0.42
TTR P02766 2/20 0.38
ALB P02768 2/20 0.38
GRM5 P41594 5/20 0.36
XDH P47989 1/20 0.36
KCNH2 Q12809 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
PGR P06401 1/20 0.32
VCAM1 P19320 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1311173 0.82 TTR (0.40) ALDH1A1CYP2A6TTRALBMEN1
SCHEMBL501406 0.82 ALDH1A1 (0.52) ALDH1A1CYP2A6TTRALBGRM5
SCHEMBL1004620 0.82 ALDH1A1 (0.52) ALDH1A1CYP2A6TTRALBGRM5
SCHEMBL16962561 0.76 ALDH1A1 (0.42) ALDH1A1CYP2A6TTRALBGRM5
SCHEMBL16950941 0.73 TTR (0.44) TTRALBMEN1KMT2APGR
SCHEMBL2811957 0.73
SCHEMBL395943 0.73
SCHEMBL2160734 0.71 ALDH1A1 (0.42) ALDH1A1CYP2A6TTRALBGRM5
SCHEMBL16958078 0.71 GRM5 (0.37) TTRALBGRM5KCNH2MEN1
SCHEMBL18934332 0.71 ALDH1A1 (0.42) ALDH1A1CYP2A6TTRALBGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900645-A1 3-PHENYLISOXAZOLIN DERIVATIVES WITH HERBICIDAL ACTION Bayer CropScience AG (DE) 2015-08-05 EP disclosed
US-6689771-B2 TREATMENT OF RHEUMATOID ARTHRITIS, OSTEOARTHRITIS, PERIODONTITIS, GINGIVITIS, CORNEAL ULCERATION, SOLID TUMOR GROWTH BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-02-10 US disclosed
US-6376665-B1 ANTIARTHRITIC AGENTS, ANTIINFLAMMATORY AGENTS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2002-04-23 US disclosed
EP-1165500-A1 AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES,TNF-ALPHA,AND AGGRECANASE Du Pont Pharmaceuticals Company (US) 2002-01-02 EP disclosed
WO-2000059874-A1 NOVEL AMIDE DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES, TNF-α, AND AGGRECANASE DU PONT PHARMACEUTICALS COMPANY (US) 2000-10-12 WO disclosed