SCHEMBL6743648

SCHEMBL6743648

Cc1ccc(C2=CCC=C2c2cc(F)c(S(C)(=O)=O)cc2F)cc1F

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.40
AKR1C3 P42330 2/20 0.36
AKR1C2 P52895 2/20 0.36
AKR1B10 O60218 1/20 0.36
AKR1C4 P17516 1/20 0.36
AKR1C1 Q04828 1/20 0.36
PTGS1 P23219 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
HSD11B1 P28845 1/20 0.33
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6746028 0.92 PTGS2 (0.49) PTGS2PTGS1NR1H2NR1H3
SCHEMBL6746854 0.90 PTGS2 (0.49) PTGS2PTGS1PDE3BPDE3ANR1H2
SCHEMBL6744855 0.90 PTGS2 (0.41) PTGS2PTGS1ALOX5APFEN1
SCHEMBL6750053 0.89 PTGS2 (0.38) PTGS2PTGS1NR1H2NR1H3
SCHEMBL6747149 0.89 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL6745224 0.87 NR1H2 (0.40) PTGS2PDE3BPDE3ANR1H2NR1H3
SCHEMBL6747140 0.87 PTGS2 (0.36) PTGS2NR1H2NR1H3ALOX5APFEN1
SCHEMBL6743170 0.87 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL6743703 0.86 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL6744624 0.86 PTGS2 (0.38) PTGS2PTGS1NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6699884-B2 ANTIINFLAMMATORY CYCLOOXYGENASE INHIBITORS. PHARMACIA CORPORATION 2004-03-02 US claimed
US-6699884-B2 ANTIINFLAMMATORY CYCLOOXYGENASE INHIBITORS. PHARMACIA CORPORATION 2004-03-02 US disclosed