SCHEMBL675763

SCHEMBL675763

CN(C)c1ccc(C(=O)NCCCCCCC(=O)NO)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 19/20 1.00
HDAC1 Q13547 13/20 1.00
HDAC2 Q92769 12/20 1.00
HDAC10 Q969S8 12/20 1.00
HDAC8 Q9BY41 11/20 1.00
HDAC3 O15379 10/20 1.00
HDAC4 P56524 9/20 1.00
HDAC7 Q8WUI4 9/20 1.00
HDAC11 Q96DB2 9/20 1.00
HDAC9 Q9UKV0 9/20 1.00
HDAC5 Q9UQL6 9/20 1.00
LTA4H P09960 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14861225 1.00 HDAC6 (1.00) HDAC6HDAC1HDAC2HDAC10HDAC8
SCHEMBL1232527 1.00 HDAC6 (1.00) HDAC6HDAC1HDAC2HDAC10HDAC8
SCHEMBL13039726 0.99 HDAC6 (0.97) HDAC6HDAC1HDAC2HDAC10HDAC8
SCHEMBL12672623 0.94 HDAC6 (0.89) HDAC6HDAC1HDAC2HDAC10HDAC8
SCHEMBL16112746 0.93 HDAC6 (0.86) HDAC6HDAC1HDAC2HDAC10HDAC8
SCHEMBL17457489 0.93 HDAC6 (0.86) HDAC6HDAC1HDAC2HDAC10HDAC8
SCHEMBL14883307 0.89 HDAC6 (0.80) HDAC6HDAC1HDAC2HDAC10HDAC8
SCHEMBL13786320 0.86 HDAC6 (0.76) HDAC6HDAC1HDAC2HDAC10HDAC8
SCHEMBL366802 0.86 HDAC6 (0.76) HDAC6HDAC1HDAC2HDAC10HDAC8
SCHEMBL28215370 0.86 HDAC6 (0.76) HDAC6HDAC1HDAC2HDAC10HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 305 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4705491-A2 SMALL MOLECULE ENHANCERS FOR ADENO-ASSOCIATED VIRUS PRODUCTION Mirus Bio LLC (US) 2026-03-11 EP claimed
EP-3350313-B1 DERIVATION OF LIVER ORGANOIDS FROM HUMAN PLURIPOTENT STEM CELLS AGENCY FOR SCIENCE TECH AND RESEARCH ASTARSTAR (SG) 2025-11-26 EP claimed
WO-2024229131-A9 SMALL MOLECULE ENHANCERS FOR ADENO-ASSOCIATED VIRUS PRODUCTION MIRUS BIO LLC (US) 2024-12-26 WO claimed
US-20240417743-A1 METHODS FOR IMPROVING GENOME ENGINEERING AND REGENERATION IN PLANT KWS SAAT SE & Co. KGaA (DE) 2024-12-19 US claimed
WO-2024229131-A2 SMALL MOLECULE ENHANCERS FOR ADENO-ASSOCIATED VIRUS PRODUCTION MIRUS BIO LLC (US) 2024-11-07 WO claimed
EP-3597705-B1 WATER ABSORBENT RESIN COMPOSITION, ABSORBENT, AND ABSORBENT ARTICLE SUMITOMO SEIKA CHEMICALS (JP) 2022-08-03 EP claimed
EP-3967323-A2 HIV VACCINE Bionor Immuno AS (NO) 2022-03-16 EP claimed
US-20200199538-A1 DERIVATION OF LIVER ORGANOIDS FROM HUMAN PLURIPOTENT STEM CELLS AGENCY FOR SCIENCE TECH AND RESEARCH ASTARSTAR (SG) 2020-06-25 US claimed
US-20200030482-A1 WATER ABSORBENT RESIN COMPOSITION, ABSORBENT, AND ABSORBENT ARTICLE SUMITOMO SEIKA CHEMICALS (JP) 2020-01-30 US claimed
CN-110582564-A derivation of liver organoids from human pluripotent stem cells 新加坡科技研究局 2019-12-17 CN claimed
WO-2011112623-A1 THIOXANTHONE-BASED AUTOPHAGY INHIBITOR THERAPIES TO TREAT CANCER SPECTRUM PHARMACEUTICALS, INC. (US) 2011-09-15 WO claimed
EP-2195029-A2 TREATMENT AND PREVENTION OF NEURODEGENERATIVE DISEASES Oryzon Genomics SA (ES) 2010-06-16 EP claimed
US-20100056522-A1 INTRAOCULAR PRESSURE-LOWERING AGENT COMPRISING COMPOUND HAVING HISTONE DEACETYLASE INHIBITOR EFFECT AS ACTIVE INGREDIENT SANTEN PHARMACEUTICAL CO., LTD. (JP) 2010-03-04 US claimed
EP-2135620-A1 OCULAR HYPOTENSIVE AGENT COMPRISING COMPOUND CAPABLE OF INHIBITING HISTONE DEACETYLASE AS ACTIVE INGREDIENT Santen Pharmaceutical Co., Ltd (JP) 2009-12-23 EP claimed
WO-2009027349-A2 TREATMENT AND PREVENTION OF NEURODEGENERATIVE DISEASES ORYZON GENOMICS SA (ES) 2009-03-05 WO claimed
WO-2008090534-A1 METHODS AND COMPOSITIONS FOR INHIBITION OF EXCESSIVE WEIGHT GAIN, REDUCTION OF INAPPROPRIATE EATING BEHAVIOURS AND INHIBITION OF BINGE EATING FOR THE TREATMENT OF OBESITY BERAND LIMITED (IE) 2008-07-31 WO claimed
WO-2007049262-A1 Methods and compositions for the promotion of neuronal growth and the treatment of asociality and affective disorders BERAND LIMITED (IE) 2007-05-03 WO claimed
US-20060148684-A1 Use of a histone deacetylase inhibitor for treating muscular dystrophies CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE-CNRS (FR) 2006-07-06 US claimed
EP-1565175-A1 USE OF A HISTONE DEACETYLASE INHIBITOR FOR TREATING MUSCULAR DYSTROPHIES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2005-08-24 EP claimed
WO-2004050076-A1 USE OF A HISTONE DEACETYLASE INHIBITOR FOR TREATING MUSCULAR DYSTROPHIES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE CNRS (FR) 2004-06-17 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100056522-A1 INTRAOCULAR PRESSURE-LOWERING AGENT COMPRISING COMPOUND HAVING HISTONE DEACETYLASE INHIBITOR EFFECT AS ACTIVE INGREDIENT HDAC1, HDAC9, HDAC5 HDAC6 10/4885HDAC1 1/4885HDAC2 8/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.