SCHEMBL6760653

SCHEMBL6760653

c1ccc(CCCCn2ccnn2)cc1

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.61
SIGMAR1 Q99720 5/20 0.45
FAAH O00519 1/20 0.45
MGLL Q99685 1/20 0.45
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
CCR3 P51677 1/20 0.44
ATP4A P20648 1/20 0.43
ATP4B P51164 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAOA P21397 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30168324 0.98 CYP19A1 (0.59) CYP19A1SIGMAR1FAAHMGLLGSK3A
SCHEMBL3113486 0.95 CYP19A1 (0.62) CYP19A1SIGMAR1GSK3AGSK3BATP4A
SCHEMBL6760657 0.87 CYP19A1 (0.67) CYP19A1MGLLGSK3AGSK3BATP4A
SCHEMBL6582554 0.86 HMOX1 (0.53) CYP19A1MGLLATP4AATP4B
SCHEMBL22398206 0.83 CYP19A1 (0.41) CYP19A1ATP4AATP4B
SCHEMBL4856182 0.83 MAOB (0.46) CYP19A1SIGMAR1MAOA
SCHEMBL2749688 0.83 CYP19A1 (0.45) CYP19A1MGLL
SCHEMBL22398040 0.83 HMOX1 (0.55) CYP19A1
SCHEMBL6580252 0.81 HMOX1 (0.54) CYP19A1MGLLATP4AATP4B
SCHEMBL22398032 0.80 ERBB2 (0.45) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111886234-A Heterocyclic mitochondrial activity inhibitors and uses thereof 蒙特利尔大学 2020-11-03 CN disclosed
US-20040106803-A1 Production method of 1-substituted-1,2,3-triazole derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-06-03 US disclosed
US-6743924-B2 EFFICIENT, HIGH YEILD SYNTHESIS OF TYROSINE KINASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-06-01 US disclosed
EP-1310491-A1 METHOD FOR PRODUCING 1-SUBSTITUTED-1,2,3-TRIAZOLE DERIVATIVE Takeda Chemical Industries, Ltd. (JP) 2003-05-14 EP disclosed
US-20030069419-A1 Method for producing 1-substituted-1,2,3- triazole derivative TAKEDA PHARMACEUTICAL COMPANY, LIMITED (JP) 2003-04-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040106803-A1 Production method of 1-substituted-1,2,3-triazole derivatives ABL1, ROS1, ADH1A CYP19A1 647/4885SIGMAR1 1646/4885FAAH 2660/4885
US-20030069419-A1 Method for producing 1-substituted-1,2,3- triazole derivative ABL1, YES1, MAP3K1 CYP19A1 686/4885SIGMAR1 1781/4885FAAH 2639/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.