SCHEMBL6760896

SCHEMBL6760896

Nc1nc(-c2ccccn2)ncc1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
ALOX15 P16050 1/20 0.47
NAPRT Q6XQN6 1/20 0.47
KDM6B O15054 1/20 0.46
KDM4A O75164 1/20 0.46
KDM5C P41229 1/20 0.46
KDM4C Q9H3R0 1/20 0.46
KDM2A Q9Y2K7 1/20 0.46
KDM3A Q9Y4C1 1/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
ALDH1A1 P00352 2/20 0.46
TP53 P04637 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MAPT P10636 1/20 0.46
GRM5 P41594 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
DHODH Q02127 1/20 0.45
HPGDS O60760 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22573444 0.85 PRKCI (0.58) ALDH1A1TDP1F2F12
SCHEMBL2558755 0.83 KDM4E (0.47) KDM4EL3MBTL1KDM6BKDM4AKDM5C
SCHEMBL30525582 0.83 KDM4E (0.47) KDM4EL3MBTL1KDM6BKDM4AKDM5C
SCHEMBL24787419 0.83 SMN1; SMN2 (0.51) KDM4EL3MBTL1ALOX15NPC1RAB9A
SCHEMBL22573273 0.83 HPGDS (0.47) KDM4EL3MBTL1ALOX15NPC1RAB9A
SCHEMBL22574062 0.82 GRM5 (0.54) KDM4EL3MBTL1NPC1RAB9ATP53
SCHEMBL3220326 0.82 HPGDS (0.51) KDM4EL3MBTL1KDM6BKDM4AKDM5C
SCHEMBL5264050 0.81 ALDH1A1 (0.65) KDM4ENPC1RAB9AALDH1A1TP53
Hydrochloric Acid SCHEMBL3217961 0.81 HPGDS (0.50) KDM4EL3MBTL1KDM6BKDM4AKDM5C
SCHEMBL22573429 0.81 HPGDS (0.67) HPGDSGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6759412-B2 FOR PRODUCING DRUGS USED FOR THERAPY OF CARDIOVASCULAR DISEASES, STABLE OR UNSTABLE ANGINA PECTORIS, CORONARY HEART DISEASE, PRINZMETAL ANGINA, ACUTE CORONARY SYNDROME, HEART FAILURE, MYOCARDIAL INFARCTION, STROKE, THROMBOSIS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2004-07-06 US disclosed