SCHEMBL6763134

SCHEMBL6763134

COc1ccc(C2=NN(C(=O)c3cccc(NC(=O)c4ccc(NC(=O)c5ccc([N+](=O)[O-])cc5)cc4)c3)CCC2)cc1OCCN(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 6/20 0.48
PGR P06401 3/20 0.46
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
PTGS2 P35354 2/20 0.43
HTR1D P28221 2/20 0.43
HTR1B P28222 2/20 0.43
HTR2A P28223 2/20 0.43
KDM4E B2RXH2 1/20 0.43
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
ALOX15 P16050 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6579233 0.91 PGR (0.49) PGRMEN1KMT2AALDH1A1CYP2C9
Dimethylamine SCHEMBL6763137 0.90 PGR (0.47) PGRMEN1KMT2AALDH1A1CYP2C9
SCHEMBL6583352 0.90 PGR (0.50) PGRMEN1KMT2AALDH1A1CYP2C9
SCHEMBL6584769 0.89 PGR (0.50) PGRMEN1KMT2AALDH1A1CYP2C9
SCHEMBL6584768 0.89 KMT2A (0.49) PGRMEN1KMT2AALDH1A1CYP2C9
SCHEMBL6583317 0.88 PGR (0.49) PGRMEN1KMT2AALDH1A1CYP2C9
SCHEMBL6763131 0.87 PGR (0.46) PGRMEN1KMT2AALDH1A1CYP2C9
SCHEMBL6582141 0.87 SETD7 (0.51) PGRMEN1KMT2AALDH1A1CYP2C9
SCHEMBL6581786 0.86 PDE4B (0.49) PGRMEN1KMT2AALDH1A1CYP2C9
SCHEMBL6578966 0.85 PGR (0.55) PGRMEN1KMT2AALDH1A1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696446-B1 HETEROCYLCIC AMIDES SUCH AS N-(4-(3-(3-(3-ETHOXY-4-METHOXY PHENYL)-1,4,5,6-TETRAHYDRO-1-PYRIDAZINYLCARBONYL)PHENYLAMINO -CARBONYL)PHENYL)-4-NITROBENZAMIDE, SUED AS PHOSPHODIESTERASE INHIBITORSFOR PROPHYLAXIS OF ALLERGIES OR ASTHMA MERCK PATENT GMBH (DE) 2004-02-24 US disclosed