SCHEMBL6764476

SCHEMBL6764476

NC(=O)C(=O)c1cc[nH]c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 1/20 0.42
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.34
MAPT P10636 2/20 0.31
POLB P06746 1/20 0.31
CYP3A4 P08684 1/20 0.31
PARP1 P09874 1/20 0.31
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31
RECQL P46063 1/20 0.31
BLM P54132 1/20 0.31
PMP22 Q01453 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PADI4 Q9UM07 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL368170 0.81
Hydrochloric Acid SCHEMBL28139048 0.79 CAPN1 (0.44) CAPN1ALDH1A1KMT2ASIRT2MAPT
Hydrochloric Acid SCHEMBL3263820 0.79
SCHEMBL28303337 0.79
SCHEMBL9528563 0.75 ALDH1A1 (0.43) CAPN1ALDH1A1KMT2ASIRT2MAPT
SCHEMBL2889586 0.73
SCHEMBL153032 0.73
Methylamine SCHEMBL27486107 0.73 ALDH1A1 (0.47) CAPN1ALDH1A1KMT2ATSHR
SCHEMBL9584944 0.72 SIRT2 (0.35) CAPN1ALDH1A1KMT2ASIRT2MAPT
SCHEMBL5158782 0.72 CAPN1 (0.47) CAPN1ALDH1A1KMT2ASIRT2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6730694-B1 SPLA2 IS A RATE LIMITING ENZYME IN THE ARACHIDONIC ACID CASCADE WHICH HYDROLYZES MEMBRANE PHOSPHOLIPIDS; TREATMENT OF SEPSIS OR RHEUMATOID ARTHRITIS ELI LILLY AND COMPANY 2004-05-04 US disclosed
EP-1307461-A2 SUBSTITUTED PYRROLE COMPOUNDS AND THEIR USE AS SPLA2 INHIBITORS ELI LILLY AND COMPANY (US) 2003-05-07 EP disclosed
WO-2002012249-A2 SUBSTITUTED PYRROLE COMPOUNDS AND THEIR USE AS SPLA2 INHIBITORS ELI LILLY AND COMPANY (US) 2002-02-14 WO disclosed